| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Lysophosphatidic acid receptor 4 |
|---|
| Ligand | BDBM50148348 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | ChEMBL_1451391 (CHEMBL3363675) |
|---|
| EC50 | 260±n/a nM |
|---|
| Citation |  Patil, R; Fells, JI; Szabó, E; Lim, KG; Norman, DD; Balogh, A; Patil, S; Strobos, J; Miller, DD; Tigyi, GJ Design and synthesis of sulfamoyl benzoic acid analogues with subnanomolar agonist activity specific to the LPA2 receptor. J Med Chem57:7136-40 (2014) [PubMed] Article |
|---|
| More Info.: | Get all data from this article, Assay Method |
|---|
| |
| Lysophosphatidic acid receptor 4 |
|---|
| Name: | Lysophosphatidic acid receptor 4 |
|---|
| Synonyms: | G-protein coupled receptor 23 | Gpr23 | Gpr23 | LPA receptor 4 | LPA-4 | LPAR4_MOUSE | Lpa4 | Lpar4 | Lysophosphatidic acid receptor 4 | P2Y purinoceptor 9 | P2y9 | Purinergic receptor 9 |
|---|
| Type: | PROTEIN |
|---|
| Mol. Mass.: | 41914.38 |
|---|
| Organism: | Mus musculus |
|---|
| Description: | ChEMBL_109462 |
|---|
| Residue: | 370 |
|---|
| Sequence: | MGDRRFIDFQFQDLNSSLRPRLGNATANNTCIVDDSFKYNLNGAVYSVVFILGLITNSAS
LFVFCFRMKMRSETAIFITNLALSDLLFVCTLPFKIFYNFNRHWPFGDTLCKISGTAFLT
NIYGSMLFLTCISVDRFLAIVYPFRSRTIRTRRNSAIVCAGVWILVLSGGISASLFSTTN
VNNATTTCFEGFSKRVWKTYLSKITIFIEVVGFIIPLILNVSCSSVVLRTLRKPATLSQI
GTNKKKVLKMITVHMAVFVVCFVPYNSVLFLYALVRSQAITNCLLERFAKIMYPITLCLA
TLNCCFDPFIYYFTLESFQKSFYINTHIRMESLFKTETPLTPKPSLPAIQEEVSDQTTNN
GGELMLESTF
|
|
|
|---|
| BDBM50148348 |
|---|
| n/a |
|---|
| Name | BDBM50148348 |
|---|
| Synonyms: | (R)-Octadec-9-enoic acid 2-hydroxy-3-phosphonooxy-propyl ester | 1-oleoyl lysophosphatidic acid | CHEMBL117021 | lysophosphatidic acid |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C21H41O7P |
|---|
| Mol. Mass. | 436.5198 |
|---|
| SMILES | CCCCCCCC\C=C/CCCCCCCC(=O)OC[C@@H](O)COP(O)(O)=O |
|---|
| Structure | 
|
|---|
Search and Browse
