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TargetCannabinoid receptor 2
LigandBDBM50058508
Substrate/Competitorn/a
Meas. Tech.ChEMBL_1459580
Ki 5.1±n/a nM
Citation Pinna GCurzu MMDore ALazzari PRuiu SPau AMurineddu GPinna GA Tricyclic pyrazoles part 7. Discovery of potent and selective dihydrothienocyclopentapyrazole derived CB2 ligands. Eur J Med Chem 85:747-57 (2014) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Cannabinoid receptor 2
Name:Cannabinoid receptor 2
Synonyms:CANNABINOID CB2 | CB-2 | CB2 | CNR2 | Cannabinoid CB2 receptor | Cannabinoid receptor | mCB2
Type:Enzyme Catalytic Domain
Mol. Mass.:38220.43
Organism:MOUSE
Description:P47936
Residue:347
Sequence:
MEGCRETEVTNGSNGGLEFNPMKEYMILSSGQQIAVAVLCTLMGLLSALENMAVLYIILS
SRRLRRKPSYLFISSLAGADFLASVIFACNFVIFHVFHGVDSNAIFLLKIGSVTMTFTAS
VGSLLLTAVDRYLCLCYPPTYKALVTRGRALVALCVMWVLSALISYLPLMGWTCCPSPCS
ELFPLIPNDYLLGWLLFIAILFSGIIYTYGYVLWKAHRHVATLAEHQDRQVPGIARMRLD
VRLAKTLGLVLAVLLICWFPALALMGHSLVTTLSDQVKEAFAFCSMLCLVNSMVNPIIYA
LRSGEIRSAAQHCLIGWKKYLQGLGPEGKEEGPRSSVTETEADVKTT
Blast this sequence in BindingDB or PDB
  Blast E-value cutoff:
BDBM50058508
n/a
NameBDBM50058508
Synonyms:CHEMBL3331460
TypeSmall organic molecule
Emp. Form.C26H29Cl2N3OS
Mol. Mass.502.499
SMILESCC(C)[C@H]1CC[C@H](C)CC1NC(=O)c1nn(c-2c1Cc1sc(C)cc-21)-c1ccc(Cl)cc1Cl |r|
Structure
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