| Reaction Details |
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 | Report a problem with these data |
| Target | Cannabinoid receptor 2 |
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| Ligand | BDBM50058501 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_1459580 (CHEMBL3369615) |
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| Ki | 5.3±n/a nM |
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| Citation |  Pinna, G; Curzu, MM; Dore, A; Lazzari, P; Ruiu, S; Pau, A; Murineddu, G; Pinna, GA Tricyclic pyrazoles part 7. Discovery of potent and selective dihydrothienocyclopentapyrazole derived CB2 ligands. Eur J Med Chem85:747-57 (2014) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Cannabinoid receptor 2 |
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| Name: | Cannabinoid receptor 2 |
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| Synonyms: | CANNABINOID CB2 | CB-2 | CB2 | CNR2_MOUSE | Cannabinoid CB2 receptor | Cannabinoid receptor | Cannabinoid receptor 2 | Cnr2 | mCB2 |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 38220.43 |
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| Organism: | MOUSE |
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| Description: | P47936 |
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| Residue: | 347 |
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| Sequence: | MEGCRETEVTNGSNGGLEFNPMKEYMILSSGQQIAVAVLCTLMGLLSALENMAVLYIILS
SRRLRRKPSYLFISSLAGADFLASVIFACNFVIFHVFHGVDSNAIFLLKIGSVTMTFTAS
VGSLLLTAVDRYLCLCYPPTYKALVTRGRALVALCVMWVLSALISYLPLMGWTCCPSPCS
ELFPLIPNDYLLGWLLFIAILFSGIIYTYGYVLWKAHRHVATLAEHQDRQVPGIARMRLD
VRLAKTLGLVLAVLLICWFPALALMGHSLVTTLSDQVKEAFAFCSMLCLVNSMVNPIIYA
LRSGEIRSAAQHCLIGWKKYLQGLGPEGKEEGPRSSVTETEADVKTT
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| BDBM50058501 |
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| n/a |
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| Name | BDBM50058501 |
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| Synonyms: | CHEMBL3331453 |
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| Type | Small organic molecule |
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| Emp. Form. | C26H27Cl2N3OS |
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| Mol. Mass. | 500.483 |
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| SMILES | Cc1csc2Cc3c(nn(c3-c12)-c1ccc(Cl)cc1Cl)C(=O)NC1[C@@]2(C)CCC(C2)C1(C)C |r,THB:22:23:26.27:29| |
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| Structure | 
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