Ki Summary new BindingDB logo
myBDB logout
Reaction Details
Report a problem with these data
TargetFormyl peptide receptor-related sequence 1
LigandBDBM50097569
Substrate/Competitorn/a
Meas. Tech.ChEMBL_1504350
EC50 2300±n/a nM
Citation Lacivita ESchepetkin IAStama MLKirpotina LNColabufo NAPerrone RKhlebnikov AIQuinn MTLeopoldo M Novel 3-(1H-indol-3-yl)-2-[3-(4-methoxyphenyl)ureido]propanamides as selective agonists of human formyl-peptide receptor 2. Bioorg Med Chem 23:3913-24 (2015) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Formyl peptide receptor-related sequence 1
Name:Formyl peptide receptor-related sequence 1
Synonyms:FMLP-R-I | FMLP-related receptor I | Formyl peptide receptor related sequence 1 | Formyl peptide receptor-like 1 | Fpr-s1 | Fpr2 | Fpr3 | Fprl1 | LXA4 receptor | Lipoxin A4 receptor | Lxa4r | N-formyl peptide receptor 2 | N-formyl peptide receptor 3
Type:PROTEIN
Mol. Mass.:39532.25
Organism:Mus musculus
Description:ChEMBL_109574
Residue:351
Sequence:
METNYSIPLNGSDVVIYDSTISRVLWILSMVVVSITFFLGVLGNGLVIWVAGFRMPHTVT
TIWYLNLALADFSFTATLPFLLVEMAMKEKWPFGWFLCKLVHIAVDVNLFGSVFLIAVIA
LDRCICVLHPVWAQNHRTVSLARNVVVGSWIFALILTLPLFLFLTTVRDARGDVHCRLSF
VSWGNSVEERLNTAITFVTTRGIIRFIVSFSLPMSFVAICYGLITTKIHKKAFVNSSRPF
RVLTGVVASFFICWFPFQLVALLGTVWLKEMQFSGSYKIIGRLVNPTSSLAFFNSCLNPI
LYVFMGQDFQERLIHSLSSRLQRALSEDSGHISDTRTNLASLPEDIEIKAI
Blast this sequence in BindingDB or PDB
  Blast E-value cutoff:
BDBM50097569
n/a
NameBDBM50097569
Synonyms:CHEMBL3590075
TypeSmall organic molecule
Emp. Form.C32H35FN4O3
Mol. Mass.542.6437
SMILESCOc1ccc(NC(=O)N[C@@H](Cc2c[nH]c3ccccc23)C(=O)NCC2(CCCCC2)c2ccc(F)cc2)cc1 |r|
Structure
Search PDB for entries with ligand similarity:Similarity to this molecule at least: