| Reaction Details |
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 | Report a problem with these data |
| Target | Formyl peptide receptor-related sequence 1 |
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| Ligand | BDBM50097565 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_1504350 (CHEMBL3592687) |
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| EC50 | 1700±n/a nM |
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| Citation |  Lacivita, E; Schepetkin, IA; Stama, ML; Kirpotina, LN; Colabufo, NA; Perrone, R; Khlebnikov, AI; Quinn, MT; Leopoldo, M Novel 3-(1H-indol-3-yl)-2-[3-(4-methoxyphenyl)ureido]propanamides as selective agonists of human formyl-peptide receptor 2. Bioorg Med Chem23:3913-24 (2015) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Formyl peptide receptor-related sequence 1 |
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| Name: | Formyl peptide receptor-related sequence 1 |
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| Synonyms: | FMLP-R-I | FMLP-related receptor I | FPRS1_MOUSE | Formyl peptide receptor related sequence 1 | Formyl peptide receptor-like 1 | Fpr-s1 | Fpr2 | Fpr3 | Fprl1 | LXA4 receptor | Lipoxin A4 receptor | Lxa4r | N-formyl peptide receptor 2 | N-formyl peptide receptor 3 |
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| Type: | PROTEIN |
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| Mol. Mass.: | 39532.25 |
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| Organism: | Mus musculus |
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| Description: | ChEMBL_109574 |
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| Residue: | 351 |
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| Sequence: | METNYSIPLNGSDVVIYDSTISRVLWILSMVVVSITFFLGVLGNGLVIWVAGFRMPHTVT
TIWYLNLALADFSFTATLPFLLVEMAMKEKWPFGWFLCKLVHIAVDVNLFGSVFLIAVIA
LDRCICVLHPVWAQNHRTVSLARNVVVGSWIFALILTLPLFLFLTTVRDARGDVHCRLSF
VSWGNSVEERLNTAITFVTTRGIIRFIVSFSLPMSFVAICYGLITTKIHKKAFVNSSRPF
RVLTGVVASFFICWFPFQLVALLGTVWLKEMQFSGSYKIIGRLVNPTSSLAFFNSCLNPI
LYVFMGQDFQERLIHSLSSRLQRALSEDSGHISDTRTNLASLPEDIEIKAI
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| BDBM50097565 |
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| n/a |
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| Name | BDBM50097565 |
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| Synonyms: | CHEMBL3589947 |
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| Type | Small organic molecule |
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| Emp. Form. | C31H34FN5O3 |
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| Mol. Mass. | 543.6318 |
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| SMILES | COc1ccc(NC(=O)N[C@@H](Cc2c[nH]c3ccccc23)C(=O)NCC2(CCCCC2)c2ccnc(F)c2)cc1 |r| |
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| Structure | 
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