| Reaction Details |
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 | Report a problem with these data |
| Target | Cannabinoid receptor 2 |
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| Ligand | BDBM50111517 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_1510274 (CHEMBL3606870) |
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| Ki | 0.600000±n/a nM |
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| Citation |  Presley, CS; Mustafa, SM; Abidi, AH; Moore, BM Synthesis and biological evaluation of (3',5'-dichloro-2,6-dihydroxy-biphenyl-4-yl)-aryl/alkyl-methanone selective CB2 inverse agonist. Bioorg Med Chem23:5390-401 (2015) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Cannabinoid receptor 2 |
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| Name: | Cannabinoid receptor 2 |
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| Synonyms: | CANNABINOID CB2 | CB-2 | CB2 | CNR2_MOUSE | Cannabinoid CB2 receptor | Cannabinoid receptor | Cannabinoid receptor 2 | Cnr2 | mCB2 |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 38220.43 |
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| Organism: | MOUSE |
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| Description: | P47936 |
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| Residue: | 347 |
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| Sequence: | MEGCRETEVTNGSNGGLEFNPMKEYMILSSGQQIAVAVLCTLMGLLSALENMAVLYIILS
SRRLRRKPSYLFISSLAGADFLASVIFACNFVIFHVFHGVDSNAIFLLKIGSVTMTFTAS
VGSLLLTAVDRYLCLCYPPTYKALVTRGRALVALCVMWVLSALISYLPLMGWTCCPSPCS
ELFPLIPNDYLLGWLLFIAILFSGIIYTYGYVLWKAHRHVATLAEHQDRQVPGIARMRLD
VRLAKTLGLVLAVLLICWFPALALMGHSLVTTLSDQVKEAFAFCSMLCLVNSMVNPIIYA
LRSGEIRSAAQHCLIGWKKYLQGLGPEGKEEGPRSSVTETEADVKTT
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| BDBM50111517 |
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| n/a |
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| Name | BDBM50111517 |
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| Synonyms: | CHEMBL3605054 |
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| Type | Small organic molecule |
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| Emp. Form. | C21H26Cl2O2 |
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| Mol. Mass. | 381.336 |
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| SMILES | CCCCCCC(C)(C)c1cc(O)c(c(O)c1)-c1cc(Cl)cc(Cl)c1 |
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| Structure | 
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