| Reaction Details |
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 | Report a problem with these data |
| Target | Delta-type opioid receptor |
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| Ligand | BDBM50114370 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_1511478 (CHEMBL3606827) |
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| Ki | 1.8±n/a nM |
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| Citation |  Loriga, G; Lazzari, P; Manca, I; Ruiu, S; Falzoi, M; Murineddu, G; Bottazzi, ME; Pinna, G; Pinna, GA Novel diazabicycloalkane delta opioid agonists. Bioorg Med Chem23:5527-38 (2015) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Delta-type opioid receptor |
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| Name: | Delta-type opioid receptor |
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| Synonyms: | DOR-1 | K56 | MSL-2 | OPIATE Delta | OPRD_MOUSE | Opioid receptors; mu and delta | Oprd1 |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 40577.25 |
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| Organism: | MOUSE |
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| Description: | P32300 |
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| Residue: | 372 |
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| Sequence: | MELVPSARAELQSSPLVNLSDAFPSAFPSAGANASGSPGARSASSLALAIAITALYSAVC
AVGLLGNVLVMFGIVRYTKLKTATNIYIFNLALADALATSTLPFQSAKYLMETWPFGELL
CKAVLSIDYYNMFTSIFTLTMMSVDRYIAVCHPVKALDFRTPAKAKLINICIWVLASGVG
VPIMVMAVTQPRDGAVVCMLQFPSPSWYWDTVTKICVFLFAFVVPILIITVCYGLMLLRL
RSVRLLSGSKEKDRSLRRITRMVLVVVGAFVVCWAPIHIFVIVWTLVDINRRDPLVVAAL
HLCIALGYANSSLNPVLYAFLDENFKRCFRQLCRTPCGRQEPGSLRRPRQATTRERVTAC
TPSDGPGGGAAA
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| BDBM50114370 |
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| n/a |
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| Name | BDBM50114370 |
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| Synonyms: | CHEMBL3604281 |
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| Type | Small organic molecule |
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| Emp. Form. | C29H39N3O2 |
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| Mol. Mass. | 461.6389 |
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| SMILES | CCN(CC)C(=O)c1ccc(cc1)C(N1CCC2CCC(C1)N2CC=C)c1cccc(OC)c1 |THB:13:14:22:18.19| |
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| Structure | 
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