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TargetDelta-type opioid receptor
LigandBDBM50114373
Substrate/Competitorn/a
Meas. Tech.ChEMBL_1511478
Ki 1.8±n/a nM
Citation Loriga GLazzari PManca IRuiu SFalzoi MMurineddu GBottazzi MEPinna GPinna GA Novel diazabicycloalkane delta opioid agonists. Bioorg Med Chem 23:5527-38 (2015) [PubMed]
More Info.:Get all data from this article,  Assay Method
 
Delta-type opioid receptor
Name:Delta-type opioid receptor
Synonyms:DOR-1 | K56 | MSL-2 | OPIATE Delta | OPRD1
Type:Enzyme Catalytic Domain
Mol. Mass.:40577.25
Organism:MOUSE
Description:P32300
Residue:372
Sequence:
MELVPSARAELQSSPLVNLSDAFPSAFPSAGANASGSPGARSASSLALAIAITALYSAVC
AVGLLGNVLVMFGIVRYTKLKTATNIYIFNLALADALATSTLPFQSAKYLMETWPFGELL
CKAVLSIDYYNMFTSIFTLTMMSVDRYIAVCHPVKALDFRTPAKAKLINICIWVLASGVG
VPIMVMAVTQPRDGAVVCMLQFPSPSWYWDTVTKICVFLFAFVVPILIITVCYGLMLLRL
RSVRLLSGSKEKDRSLRRITRMVLVVVGAFVVCWAPIHIFVIVWTLVDINRRDPLVVAAL
HLCIALGYANSSLNPVLYAFLDENFKRCFRQLCRTPCGRQEPGSLRRPRQATTRERVTAC
TPSDGPGGGAAA
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  Blast E-value cutoff:
BDBM50114373
n/a
NameBDBM50114373
Synonyms:CHEMBL3604278
TypeSmall organic molecule
Emp. Form.C27H35N3O2
Mol. Mass.433.5857
SMILESCCN(CC)C(=O)c1ccc(cc1)C(N1C2CC1CN(CC=C)C2)c1cccc(OC)c1 |THB:13:14:23.19.18:16|
Structure
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