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TargetP2Y purinoceptor 11
LigandBDBM50131059
Substrate/Competitorn/a
Meas. Tech.ChEBML_1526465
EC50 8700±n/a nM
Citation Azran, SDanino, OFörster, DKenigsberg, SReiser, GDixit, MSingh, VMajor, DTFischer, B Identification of Highly Promising Antioxidants/Neuroprotectants Based on Nucleoside 5'-Phosphorothioate Scaffold. Synthesis, Activity, and Mechanisms of Action. J Med Chem58:8427-43 (2015) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
P2Y purinoceptor 11
Name:P2Y purinoceptor 11
Synonyms:P2RY11 | P2Y purinoceptor 11 | P2Y11 | P2Y11_HUMAN | Purinergic receptor P2Y11
Type:PROTEIN
Mol. Mass.:40366.02
Organism:Homo sapiens (Human)
Description:ChEMBL_1362532
Residue:374
Sequence:
MAANVSGAKSCPANFLAAADDKLSGFQGDFLWPILVVEFLVAVASNGLALYRFSIRKQRP
WHPAVVFSVQLAVSDLLCALTLPPLAAYLYPPKHWRYGEAACRLERFLFTCNLLGSVIFI
TCISLNRYLGIVHPFFARSHLRPKHAWAVSAAGWVLAALLAMPTLSFSHLKRPQQGAGNC
SVARPEACIKCLGTADHGLAAYRAYSLVLAGLGCGLPLLLTLAAYGALGRAVLRSPGMTV
AEKLRVAALVASGVALYASSYVPYHIMRVLNVDARRRWSTRCPSFADIAQATAALELGPY
VGYQVMRGLMPLAFCVHPLLYMAAVPSLGCCCRHCPGYRDSWNPEDAKSTGQALPLNATA
APKPSEPQSRELSQ
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  Blast E-value cutoff:
BDBM50131059
n/a
NameBDBM50131059
Synonyms:CHEMBL575257
TypeSmall organic molecule
Emp. Form.C10H15N5O9P2S
Mol. Mass.443.267
SMILESNc1ncnc2n(cnc12)[C@@H]1O[C@H](COP(S)(=O)OP(O)(O)=O)[C@@H](O)[C@H]1O |r|
Structure
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