| Reaction Details |
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 | Report a problem with these data |
| Target | Mu-type opioid receptor |
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| Ligand | BDBM50123658 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_1552632 (CHEMBL3762571) |
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| IC50 | 1±n/a nM |
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| Citation |  Turnaturi, R; Aricò, G; Ronsisvalle, G; Parenti, C; Pasquinucci, L Multitarget opioid ligands in pain relief: New players in an old game. Eur J Med Chem108:211-28 (2016) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Mu-type opioid receptor |
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| Name: | Mu-type opioid receptor |
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| Synonyms: | M-OR-1 | MOR-1 | Mu opioid receptor | Mu-type opioid receptor (Mu) | OPIATE Mu | OPRM1 | OPRM_CAVPO |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 11165.58 |
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| Organism: | GUINEA PIG |
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| Description: | P97266 |
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| Residue: | 98 |
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| Sequence: | YTKMKTATNIYIFNLALADALATSTLPFQSVNYLMGTWPFGTILCKIVISIDYYNMFTSI
FTLCTMSVDRYIAVCHPVKALDFRTPRNAKTVNVCNWI
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|
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| BDBM50123658 |
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| n/a |
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| Name | BDBM50123658 |
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| Synonyms: | 3-[(R)-((2S,5R)-4-Allyl-2,5-dimethyl-piperazin-1-yl)-(3-hydroxy-phenyl)-methyl]-N-(3-fluoro-phenyl)-N-methyl-benzamide | CHEMBL155892 |
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| Type | Small organic molecule |
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| Emp. Form. | C30H34FN3O2 |
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| Mol. Mass. | 487.6083 |
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| SMILES | C[C@@H]1CN([C@@H](c2cccc(O)c2)c2cccc(c2)C(=O)N(C)c2cccc(F)c2)[C@@H](C)CN1CC=C |
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| Structure | 
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