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TargetG-protein coupled receptor 55
LigandBDBM50152128
Substrate/Competitorn/a
Meas. Tech.ChEMBL_1561203 (CHEMBL3777631)
IC50 770±n/a nM
Citation Meza-Aviņa, MELingerfelt, MAConsole-Bram, LMGamage, TFSharir, HGettys, KEHurst, DPKotsikorou, EShore, DMCaron, MGRao, NBarak, LSAbood, MEReggio, PHCroatt, MP Design, synthesis, and analysis of antagonists of GPR55: Piperidine-substituted 1,3,4-oxadiazol-2-ones. Bioorg Med Chem Lett26:1827-30 (2016) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
G-protein coupled receptor 55
Name:G-protein coupled receptor 55
Synonyms:G protein-coupled receptor 55 | GPR55 | GPR55_HUMAN
Type:PROTEIN
Mol. Mass.:36649.72
Organism:Homo sapiens (Human)
Description:ChEMBL_1292265
Residue:319
Sequence:
MSQQNTSGDCLFDGVNELMKTLQFAVHIPTFVLGLLLNLLAIHGFSTFLKNRWPDYAATS
IYMINLAVFDLLLVLSLPFKMVLSQVQSPFPSLCTLVECLYFVSMYGSVFTICFISMDRF
LAIRYPLLVSHLRSPRKIFGICCTIWVLVWTGSIPIYSFHGKVEKYMCFHNMSDDTWSAK
VFFPLEVFGFLLPMGIMGFCCSRSIHILLGRRDHTQDWVQQKACIYSIAASLAVFVVSFL
PVHLGFFLQFLVRNSFIVECRAKQSISFFLQLSMCFSNVNCCLDVFCYYFVIKEFRMNIR
AHRPSRVQLVLQDTTISRG
Blast this sequence in BindingDB or PDB
  Blast E-value cutoff:
BDBM50152128
n/a
NameBDBM50152128
Synonyms:CHEMBL3775187
TypeSmall organic molecule
Emp. Form.C26H29N3O3
Mol. Mass.431.5268
SMILESCc1ccc(cc1)C1(CC1(C)C)C(=O)N1CCC(CC1)n1nc(oc1=O)-c1ccccc1
Structure
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