| Reaction Details |
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 | Report a problem with these data |
| Target | Somatostatin receptor type 2 |
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| Ligand | BDBM50155306 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_1565563 (CHEMBL3782232) |
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| Ki | 4690±n/a nM |
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| Citation |  Fridén-Saxin, M; Seifert, T; Malo, M; da Silva Andersson, K; Pemberton, N; Dyrager, C; Friberg, A; Dahlén, K; Wallén, EA; Grøtli, M; Luthman, K Chroman-4-one and chromone based somatostatinß-turn mimetics. Eur J Med Chem114:59-64 (2016) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Somatostatin receptor type 2 |
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| Name: | Somatostatin receptor type 2 |
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| Synonyms: | SOMATOSTATIN SST2 | SRIF-1 | SS-2-R | SS2-R | SS2R | SSR2_HUMAN | SSTR2 | Somatostatin receptor type 2 (SSTR2) |
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| Type: | Enzyme |
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| Mol. Mass.: | 41344.94 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P30874 |
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| Residue: | 369 |
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| Sequence: | MDMADEPLNGSHTWLSIPFDLNGSVVSTNTSNQTEPYYDLTSNAVLTFIYFVVCIIGLCG
NTLVIYVILRYAKMKTITNIYILNLAIADELFMLGLPFLAMQVALVHWPFGKAICRVVMT
VDGINQFTSIFCLTVMSIDRYLAVVHPIKSAKWRRPRTAKMITMAVWGVSLLVILPIMIY
AGLRSNQWGRSSCTINWPGESGAWYTGFIIYTFILGFLVPLTIICLCYLFIIIKVKSSGI
RVGSSKRKKSEKKVTRMVSIVVAVFIFCWLPFYIFNVSSVSMAISPTPALKGMFDFVVVL
TYANSCANPILYAFLSDNFKKSFQNVLCLVKVSGTDDGERSDSKQDKSRLNETTETQRTL
LNGDLQTSI
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| BDBM50155306 |
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| n/a |
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| Name | BDBM50155306 |
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| Synonyms: | CHEMBL3781875 |
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| Type | Small organic molecule |
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| Emp. Form. | C21H26N2O2 |
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| Mol. Mass. | 338.4433 |
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| SMILES | NCCCCCOc1ccccc1OCCc1c[nH]c2ccccc12 |
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| Structure | 
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