| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Somatostatin receptor type 4 |
|---|
| Ligand | BDBM50155309 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | ChEMBL_1565560 (CHEMBL3782229) |
|---|
| Ki | 7090±n/a nM |
|---|
| Citation |  Fridén-Saxin, M; Seifert, T; Malo, M; da Silva Andersson, K; Pemberton, N; Dyrager, C; Friberg, A; Dahlén, K; Wallén, EA; Grøtli, M; Luthman, K Chroman-4-one and chromone based somatostatinß-turn mimetics. Eur J Med Chem114:59-64 (2016) [PubMed] Article |
|---|
| More Info.: | Get all data from this article, Assay Method |
|---|
| |
| Somatostatin receptor type 4 |
|---|
| Name: | Somatostatin receptor type 4 |
|---|
| Synonyms: | SOMATOSTATIN SST4 | SS-4-R | SS4-R | SS4R | SSR4_HUMAN | SST4R | SSTR4 | Somatostatin receptor type 4 (SSTR4) |
|---|
| Type: | Enzyme |
|---|
| Mol. Mass.: | 42015.38 |
|---|
| Organism: | Homo sapiens (Human) |
|---|
| Description: | P31391 |
|---|
| Residue: | 388 |
|---|
| Sequence: | MSAPSTLPPGGEEGLGTAWPSAANASSAPAEAEEAVAGPGDARAAGMVAIQCIYALVCLV
GLVGNALVIFVILRYAKMKTATNIYLLNLAVADELFMLSVPFVASSAALRHWPFGSVLCR
AVLSVDGLNMFTSVFCLTVLSVDRYVAVVHPLRAATYRRPSVAKLINLGVWLASLLVTLP
IAIFADTRPARGGQAVACNLQWPHPAWSAVFVVYTFLLGFLLPVLAIGLCYLLIVGKMRA
VALRAGWQQRRRSEKKITRLVLMVVVVFVLCWMPFYVVQLLNLFVTSLDATVNHVSLILS
YANSCANPILYGFLSDNFRRFFQRVLCLRCCLLEGAGGAEEEPLDYYATALKSKGGAGCM
CPPLPCQQEALQPEPGRKRIPLTRTTTF
|
|
|
|---|
| BDBM50155309 |
|---|
| n/a |
|---|
| Name | BDBM50155309 |
|---|
| Synonyms: | CHEMBL3780496 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C24H24ClNO2 |
|---|
| Mol. Mass. | 393.906 |
|---|
| SMILES | NCCCc1cc(Cl)cc2C(=O)CC(CCc3cccc4ccccc34)Oc12 |
|---|
| Structure | 
|
|---|
Search and Browse
