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TargetG-protein coupled receptor 55
LigandBDBM50156112
Substrate/Competitorn/a
Meas. Tech.ChEMBL_1563025 (CHEMBL3783507)
EC50 28±n/a nM
Citation Morales, PWhyte, LSChicharro, RGómez-Cañas, MPazos, MRGoya, PIrving, AJFernández-Ruiz, JRoss, RAJagerovic, N Identification of Novel GPR55 Modulators Using Cell-Impedance-Based Label-Free Technology. J Med Chem59:1840-53 (2016) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
G-protein coupled receptor 55
Name:G-protein coupled receptor 55
Synonyms:G protein-coupled receptor 55 | GPR55 | GPR55_HUMAN
Type:PROTEIN
Mol. Mass.:36649.72
Organism:Homo sapiens (Human)
Description:ChEMBL_1292265
Residue:319
Sequence:
MSQQNTSGDCLFDGVNELMKTLQFAVHIPTFVLGLLLNLLAIHGFSTFLKNRWPDYAATS
IYMINLAVFDLLLVLSLPFKMVLSQVQSPFPSLCTLVECLYFVSMYGSVFTICFISMDRF
LAIRYPLLVSHLRSPRKIFGICCTIWVLVWTGSIPIYSFHGKVEKYMCFHNMSDDTWSAK
VFFPLEVFGFLLPMGIMGFCCSRSIHILLGRRDHTQDWVQQKACIYSIAASLAVFVVSFL
PVHLGFFLQFLVRNSFIVECRAKQSISFFLQLSMCFSNVNCCLDVFCYYFVIKEFRMNIR
AHRPSRVQLVLQDTTISRG
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  Blast E-value cutoff:
BDBM50156112
n/a
NameBDBM50156112
Synonyms:CHEMBL3780748
TypeSmall organic molecule
Emp. Form.C27H33N5O4
Mol. Mass.491.582
SMILESCOc1ccc2-c3nn(CNC(=O)CN4CCN(CC4)c4ccccc4OC)cc3C(C)(C)Oc2c1
Structure
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