Reaction Details |
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Target | G-protein coupled receptor 55 |
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Ligand | BDBM50156112 |
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Substrate/Competitor | n/a |
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Meas. Tech. | ChEMBL_1563025 (CHEMBL3783507) |
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EC50 | 28±n/a nM |
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Citation | Morales, P; Whyte, LS; Chicharro, R; Gómez-Cañas, M; Pazos, MR; Goya, P; Irving, AJ; Fernández-Ruiz, J; Ross, RA; Jagerovic, N Identification of Novel GPR55 Modulators Using Cell-Impedance-Based Label-Free Technology. J Med Chem59:1840-53 (2016) [PubMed] Article |
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More Info.: | Get all data from this article, Assay Method |
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G-protein coupled receptor 55 |
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Name: | G-protein coupled receptor 55 |
Synonyms: | G protein-coupled receptor 55 | GPR55 | GPR55_HUMAN |
Type: | PROTEIN |
Mol. Mass.: | 36649.72 |
Organism: | Homo sapiens (Human) |
Description: | ChEMBL_1292265 |
Residue: | 319 |
Sequence: | MSQQNTSGDCLFDGVNELMKTLQFAVHIPTFVLGLLLNLLAIHGFSTFLKNRWPDYAATS
IYMINLAVFDLLLVLSLPFKMVLSQVQSPFPSLCTLVECLYFVSMYGSVFTICFISMDRF
LAIRYPLLVSHLRSPRKIFGICCTIWVLVWTGSIPIYSFHGKVEKYMCFHNMSDDTWSAK
VFFPLEVFGFLLPMGIMGFCCSRSIHILLGRRDHTQDWVQQKACIYSIAASLAVFVVSFL
PVHLGFFLQFLVRNSFIVECRAKQSISFFLQLSMCFSNVNCCLDVFCYYFVIKEFRMNIR
AHRPSRVQLVLQDTTISRG
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BDBM50156112 |
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n/a |
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Name | BDBM50156112 |
Synonyms: | CHEMBL3780748 |
Type | Small organic molecule |
Emp. Form. | C27H33N5O4 |
Mol. Mass. | 491.582 |
SMILES | COc1ccc2-c3nn(CNC(=O)CN4CCN(CC4)c4ccccc4OC)cc3C(C)(C)Oc2c1 |
Structure |
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