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TargetChromobox protein homolog 7
LigandBDBM50157400
Substrate/Competitorn/a
Meas. Tech.ChEBML_1565749
Kd 34000±n/a nM
Citation Milosevich NGignac MCMcFarlane JSimhadri CHorvath SDaze KDCroft CSDheri AQuon TTDouglas SFWulff JEPaci IHof F Selective Inhibition of CBX6: A Methyllysine Reader Protein in the Polycomb Family. ACS Med Chem Lett 7:139-44 (2016) [PubMed]
More Info.:Get all data from this article,  Assay Method
 
Chromobox protein homolog 7
Name:Chromobox protein homolog 7
Synonyms:CBX7 | Chromobox protein homolog 7
Type:Protein
Mol. Mass.:28351.76
Organism:Homo sapiens (Human)
Description:n/a
Residue:251
Sequence:
MELSAIGEQVFAVESIRKKRVRKGKVEYLVKWKGWPPKYSTWEPEEHILDPRLVMAYEEK
EERDRASGYRKRGPKPKRLLLQRLYSMDLRSSHKAKGKEKLCFSLTCPLGSGSPEGVVKA
GAPELVDKGPLVPTLPFPLRKPRKAHKYLRLSRKKFPPRGPNLESHSHRRELFLQEPPAP
DVLQAAGEWEPAAQPPEEEADADLAEGPPPWTPALPSSEVTVTDITANSITVTFREAQAA
EGFFRDRSGKF
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  Blast E-value cutoff:
BDBM50157400
n/a
NameBDBM50157400
Synonyms:CHEMBL3781600
TypeSmall organic molecule
Emp. Form.C63H90BrN12O14S
Mol. Mass.1351.429
SMILES[H][C@]12CS[C@@H](CCCCC(=O)NCCCC[C@H](NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](CO)NC(=O)[C@H](CCCC[N+](C)(C)C)NC(=O)[C@H](Cc3ccc(O)cc3)NC(=O)[C@@H](NC(=O)[C@H](Cc3ccccc3)NC(=O)c3ccc(Br)cc3)C(C)C)C(N)=O)[C@@]1([H])NC(=O)N2 |r|
Structure
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