| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Inhibitor of growth protein 2 |
|---|
| Ligand | BDBM18959 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | ChEMBL_1566080 (CHEMBL3791708) |
|---|
| IC50 | 97000±n/a nM |
|---|
| Citation |  McAllister, TE; England, KS; Hopkinson, RJ; Brennan, PE; Kawamura, A; Schofield, CJ Recent Progress in Histone Demethylase Inhibitors. J Med Chem59:1308-29 (2016) [PubMed] Article |
|---|
| More Info.: | Get all data from this article, Assay Method |
|---|
| |
| Inhibitor of growth protein 2 |
|---|
| Name: | Inhibitor of growth protein 2 |
|---|
| Synonyms: | ING1L | ING1Lp | ING2 | ING2_HUMAN | Inhibitor of growth 1-like protein | Inhibitor of growth protein 2 | p32 | p33ING2 |
|---|
| Type: | PROTEIN |
|---|
| Mol. Mass.: | 32812.71 |
|---|
| Organism: | Homo sapiens (Human) |
|---|
| Description: | ChEMBL_116766 |
|---|
| Residue: | 280 |
|---|
| Sequence: | MLGQQQQQLYSSAALLTGERSRLLTCYVQDYLECVESLPHDMQRNVSVLRELDNKYQETL
KEIDDVYEKYKKEDDLNQKKRLQQLLQRALINSQELGDEKIQIVTQMLELVENRARQMEL
HSQCFQDPAESERASDKAKMDSSQPERSSRRPRRQRTSESRDLCHMANGIEDCDDQPPKE
KKSKSAKKKKRSKAKQEREASPVEFAIDPNEPTYCLCNQVSYGEMIGCDNEQCPIEWFHF
SCVSLTYKPKGKWYCPKCRGDNEKTMDKSTEKTKKDRRSR
|
|
|
|---|
| BDBM18959 |
|---|
| n/a |
|---|
| Name | BDBM18959 |
|---|
| Synonyms: | 3-{[4-(2-aminoethoxy)-3,5-diiodophenyl]carbonyl}-2-butyl-1-benzofuran | CHEMBL1598 | DDEA | Desdiethylamiodarone | Di-N-desethylamiodarone | L 33530 | Methanone |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C21H21I2NO3 |
|---|
| Mol. Mass. | 589.2053 |
|---|
| SMILES | CCCCc1oc2ccccc2c1C(=O)c1cc(I)c(OCCN)c(I)c1 |
|---|
| Structure | 
|
|---|
Search and Browse
