| Reaction Details |
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 | Report a problem with these data |
| Target | C-terminal-binding protein 2 |
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| Ligand | BDBM50167651 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_1574551 (CHEMBL3804623) |
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| IC50 | 116300±n/a nM |
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| Citation |  Korwar, S; Morris, BL; Parikh, HI; Coover, RA; Doughty, TW; Love, IM; Hilbert, BJ; Royer, WE; Kellogg, GE; Grossman, SR; Ellis, KC Design, synthesis, and biological evaluation of substrate-competitive inhibitors of C-terminal Binding Protein (CtBP). Bioorg Med Chem24:2707-15 (2016) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| C-terminal-binding protein 2 |
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| Name: | C-terminal-binding protein 2 |
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| Synonyms: | C-terminal-binding protein 2 | C-terminal-binding protein 2 (CtBP2) | CTBP2 | CTBP2_HUMAN |
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| Type: | Protein |
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| Mol. Mass.: | 48948.33 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P56545 |
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| Residue: | 445 |
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| Sequence: | MALVDKHKVKRQRLDRICEGIRPQIMNGPLHPRPLVALLDGRDCTVEMPILKDLATVAFC
DAQSTQEIHEKVLNEAVGAMMYHTITLTREDLEKFKALRVIVRIGSGYDNVDIKAAGELG
IAVCNIPSAAVEETADSTICHILNLYRRNTWLYQALREGTRVQSVEQIREVASGAARIRG
ETLGLIGFGRTGQAVAVRAKAFGFSVIFYDPYLQDGIERSLGVQRVYTLQDLLYQSDCVS
LHCNLNEHNHHLINDFTIKQMRQGAFLVNAARGGLVDEKALAQALKEGRIRGAALDVHES
EPFSFAQGPLKDAPNLICTPHTAWYSEQASLEMREAAATEIRRAITGRIPESLRNCVNKE
FFVTSAPWSVIDQQAIHPELNGATYRYPPGIVGVAPGGLPAAMEGIIPGGIPVTHNLPTV
AHPSQAPSPNQPTKHGDNREHPNEQ
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| BDBM50167651 |
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| n/a |
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| Name | BDBM50167651 |
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| Synonyms: | CHEBI:30851 | Phenylpyruvate |
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| Type | Small organic molecule |
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| Emp. Form. | C9H8O3 |
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| Mol. Mass. | 164.158 |
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| SMILES | OC(=O)C(=O)Cc1ccccc1 |
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| Structure | 
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