| Reaction Details |
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 | Report a problem with these data |
| Target | Delta-type opioid receptor |
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| Ligand | BDBM50168140 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_1575958 (CHEMBL3802787) |
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| EC50 | 158489±n/a nM |
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| Citation |  Pasquinucci, L; Turnaturi, R; Aricò, G; Parenti, C; Pallaki, P; Georgoussi, Z; Ronsisvalle, S Evaluation of N-substituent structural variations in opioid receptor profile of LP1. Bioorg Med Chem24:2832-42 (2016) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Delta-type opioid receptor |
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| Name: | Delta-type opioid receptor |
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| Synonyms: | DOR-1 | K56 | MSL-2 | OPIATE Delta | OPRD_MOUSE | Opioid receptors; mu and delta | Oprd1 |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 40577.25 |
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| Organism: | MOUSE |
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| Description: | P32300 |
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| Residue: | 372 |
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| Sequence: | MELVPSARAELQSSPLVNLSDAFPSAFPSAGANASGSPGARSASSLALAIAITALYSAVC
AVGLLGNVLVMFGIVRYTKLKTATNIYIFNLALADALATSTLPFQSAKYLMETWPFGELL
CKAVLSIDYYNMFTSIFTLTMMSVDRYIAVCHPVKALDFRTPAKAKLINICIWVLASGVG
VPIMVMAVTQPRDGAVVCMLQFPSPSWYWDTVTKICVFLFAFVVPILIITVCYGLMLLRL
RSVRLLSGSKEKDRSLRRITRMVLVVVGAFVVCWAPIHIFVIVWTLVDINRRDPLVVAAL
HLCIALGYANSSLNPVLYAFLDENFKRCFRQLCRTPCGRQEPGSLRRPRQATTRERVTAC
TPSDGPGGGAAA
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| BDBM50168140 |
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| n/a |
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| Name | BDBM50168140 |
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| Synonyms: | CHEMBL3797702 |
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| Type | Small organic molecule |
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| Emp. Form. | C26H29N3O2 |
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| Mol. Mass. | 415.5274 |
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| SMILES | [H][C@]12Cc3ccc(O)cc3[C@](C)(CCN1CCC(=O)Nc1cccc3cnccc13)[C@H]2C |r,THB:8:9:30:14.13.12,15:14:30:3.9.2| |
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| Structure | 
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