| Reaction Details |
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 | Report a problem with these data |
| Target | Mu-type opioid receptor |
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| Ligand | BDBM50142692 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEBML_1575957 |
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| EC50 | 794±n/a nM |
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| Citation |  Pasquinucci, L; Turnaturi, R; Aricò, G; Parenti, C; Pallaki, P; Georgoussi, Z; Ronsisvalle, S Evaluation of N-substituent structural variations in opioid receptor profile of LP1. Bioorg Med Chem24:2832-42 (2016) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Mu-type opioid receptor |
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| Name: | Mu-type opioid receptor |
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| Synonyms: | M-OR-1 | MOR-1 | Mu opioid receptor | Mu-type opioid receptor (Mu) | OPIATE Mu | OPRM1 | OPRM_CAVPO |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 11165.58 |
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| Organism: | GUINEA PIG |
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| Description: | P97266 |
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| Residue: | 98 |
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| Sequence: | YTKMKTATNIYIFNLALADALATSTLPFQSVNYLMGTWPFGTILCKIVISIDYYNMFTSI
FTLCTMSVDRYIAVCHPVKALDFRTPRNAKTVNVCNWI
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| BDBM50142692 |
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| n/a |
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| Name | BDBM50142692 |
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| Synonyms: | CHEMBL3759092 |
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| Type | Small organic molecule |
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| Emp. Form. | C23H28N2O2 |
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| Mol. Mass. | 364.4806 |
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| SMILES | [H][C@]12Cc3ccc(O)cc3[C@](C)(CCN1CCC(=O)Nc1ccccc1)[C@H]2C |r,THB:8:9:26:12.14.13,15:14:26:3.9.2| |
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| Structure | 
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