| Reaction Details |
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 | Report a problem with these data |
| Target | Cytosol aminopeptidase [33-68,L62W] |
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| Ligand | BDBM50170875 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_1577950 (CHEMBL3806574) |
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| Ki | 7020±n/a nM |
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| Citation |  Weglarz-Tomczak, E; Berlicki, L; Pawelczak, M; Nocek, B; Joachimiak, A; Mucha, A A structural insight into the P1S1 binding mode of diaminoethylphosphonic and phosphinic acids, selective inhibitors of alanine aminopeptidases. Eur J Med Chem117:187-96 (2016) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Cytosol aminopeptidase [33-68,L62W] |
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| Name: | Cytosol aminopeptidase [33-68,L62W] |
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| Synonyms: | AMPL_PIG | Cytosol aminopeptidase | LAP3 | Leucine aminopeptidase (LAP) |
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| Type: | Enzyme |
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| Mol. Mass.: | 4015.44 |
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| Organism: | Sus scrofa (Pig) |
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| Description: | P28839[33-68,L62W] |
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| Residue: | 36 |
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| Sequence: | TKGLVLGIYSKEKEDDAPQFTSAGENFDKWVSGKLR
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| BDBM50170875 |
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| n/a |
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| Name | BDBM50170875 |
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| Synonyms: | CHEMBL3805288 |
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| Type | Small organic molecule |
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| Emp. Form. | C9H16N3O3P |
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| Mol. Mass. | 245.2154 |
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| SMILES | NC(CNCc1ccc(N)cc1)P(O)(O)=O |
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| Structure | 
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