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TargetCytosol aminopeptidase [33-68,L62W]
LigandBDBM50170880
Substrate/Competitorn/a
Meas. Tech.ChEMBL_1577950 (CHEMBL3806574)
Ki 21000±n/a nM
Citation Weglarz-Tomczak, EBerlicki, LPawelczak, MNocek, BJoachimiak, AMucha, A A structural insight into the P1S1 binding mode of diaminoethylphosphonic and phosphinic acids, selective inhibitors of alanine aminopeptidases. Eur J Med Chem117:187-96 (2016) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Cytosol aminopeptidase [33-68,L62W]
Name:Cytosol aminopeptidase [33-68,L62W]
Synonyms:AMPL_PIG | Cytosol aminopeptidase | LAP3 | Leucine aminopeptidase (LAP)
Type:Enzyme
Mol. Mass.:4015.44
Organism:Sus scrofa (Pig)
Description:P28839[33-68,L62W]
Residue:36
Sequence:
TKGLVLGIYSKEKEDDAPQFTSAGENFDKWVSGKLR
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  Blast E-value cutoff:
BDBM50170880
n/a
NameBDBM50170880
Synonyms:CHEMBL3806187
TypeSmall organic molecule
Emp. Form.C15H25N2O4P
Mol. Mass.328.3438
SMILESCCCNCC(N)P(O)(=O)CC(Cc1ccccc1)C(O)=O
Structure
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