| Reaction Details |
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 | Report a problem with these data |
| Target | 5'-AMP-activated protein kinase subunit gamma-1 |
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| Ligand | BDBM50195534 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_1617806 (CHEMBL3859875) |
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| EC50 | 2.0±n/a nM |
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| Citation |  Cameron, KO; Kurumbail, RG Recent progress in the identification of adenosine monophosphate-activated protein kinase (AMPK) activators. Bioorg Med Chem Lett26:5139-5148 (2016) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| 5'-AMP-activated protein kinase subunit gamma-1 |
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| Name: | 5'-AMP-activated protein kinase subunit gamma-1 |
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| Synonyms: | 5'-AMP-activated protein kinase subunit gamma-1 | AAKG1_HUMAN | AMP-activated protein kinase, gamma-1 subunit | AMPK alpha2/beta2/gamma1 | AMPK gamma-1 | AMPK gamma1 | AMPK subunit gamma-1 | AMPKg | PRKAG1 |
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| Type: | n/a |
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| Mol. Mass.: | 37581.44 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P54619 |
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| Residue: | 331 |
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| Sequence: | METVISSDSSPAVENEHPQETPESNNSVYTSFMKSHRCYDLIPTSSKLVVFDTSLQVKKA
FFALVTNGVRAAPLWDSKKQSFVGMLTITDFINILHRYYKSALVQIYELEEHKIETWREV
YLQDSFKPLVCISPNASLFDAVSSLIRNKIHRLPVIDPESGNTLYILTHKRILKFLKLFI
TEFPKPEFMSKSLEELQIGTYANIAMVRTTTPVYVALGIFVQHRVSALPVVDEKGRVVDI
YSKFDVINLAAEKTYNNLDVSVTKALQHRSHYFEGVLKCYLHETLETIINRLVEAEVHRL
VVVDENDVVKGIVSLSDILQALVLTGGEKKP
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| BDBM50195534 |
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| n/a |
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| Name | BDBM50195534 |
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| Synonyms: | CHEMBL3957286 |
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| Type | Small organic molecule |
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| Emp. Form. | C25H21ClN2O6 |
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| Mol. Mass. | 480.897 |
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| SMILES | [H][C@]12OC[C@@H](Oc3nc4cc(c(Cl)cc4[nH]3)-c3ccc(cc3)-c3c(O)cccc3O)[C@@]1([H])OC[C@H]2O |r| |
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| Structure | 
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