| Reaction Details |
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 | Report a problem with these data |
| Target | Transmembrane domain-containing protein TMIGD3 |
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| Ligand | BDBM50199453 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_1621587 (CHEMBL3863870) |
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| Ki | 165±n/a nM |
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| Citation |  Tosh, DK; Ciancetta, A; Warnick, E; Crane, S; Gao, ZG; Jacobson, KA Structure-Based Scaffold Repurposing for G Protein-Coupled Receptors: Transformation of Adenosine Derivatives into 5HT J Med Chem59:11006-11026 (2016) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Transmembrane domain-containing protein TMIGD3 |
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| Name: | Transmembrane domain-containing protein TMIGD3 |
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| Synonyms: | TMIG3_HUMAN | TMIGD3 | Transmembrane domain-containing protein TMIGD3 |
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| Type: | PROTEIN |
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| Mol. Mass.: | 30335.79 |
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| Organism: | Homo sapiens (Human) |
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| Description: | ChEMBL_114868 |
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| Residue: | 266 |
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| Sequence: | MEGSPAGPIEQKEARWESSWEEQPDWTLGCLSPESQFRIPGLPGCILSFQLKVCFLPVMW
LFILLSLALISDAMVMDEKVKRSFVLDTASAICNYNAHYKNHPKYWCRGYFRDYCNIIAF
SPNSTNHVALRDTGNQLIVTMSCLTKEDTGWYWCGIQRDFARDDMDFTELIVTDDKGTLA
NDFWSGKDLSGNKTRSCKAPKVVRKADRSRTSILIICILITGLGIISVISHLTKRRRSQR
NRRVGNTLKPFSRVLTPKEMAPTEQM
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| BDBM50199453 |
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| n/a |
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| Name | BDBM50199453 |
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| Synonyms: | CHEMBL3914002 |
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| Type | Small organic molecule |
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| Emp. Form. | C12H9Cl2N5 |
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| Mol. Mass. | 294.139 |
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| SMILES | Clc1cccc(CNc2nc(Cl)nc3[nH]cnc23)c1 |
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| Structure | 
|
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