| Reaction Details |
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 | Report a problem with these data |
| Target | D(3) dopamine receptor |
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| Ligand | BDBM50207049 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_1629511 (CHEMBL3872137) |
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| Ki | 126±n/a nM |
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| Citation |  Saavedra, OM; Karila, D; Brossard, D; Rojas, A; Dupuis, D; Gohier, A; Mannoury la Cour, C; Millan, MJ; Ortuno, JC; Hanessian, S Design and synthesis of novel N-sulfonyl-2-indoles that behave as 5-HT Bioorg Med Chem25:38-52 (2017) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| D(3) dopamine receptor |
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| Name: | D(3) dopamine receptor |
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| Synonyms: | DOPAMINE D3 | DRD3 | DRD3_HUMAN | Dopamine D3 receptor | Dopamine D3 receptor (D3) | Dopamine D3 receptor (D3R) | Dopamine receptor | Dopamine receptor (D3) | Dopamine receptor D3 |
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| Type: | n/a |
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| Mol. Mass.: | 44243.43 |
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| Organism: | Homo sapiens (Human) |
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| Description: | n/a |
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| Residue: | 400 |
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| Sequence: | MASLSQLSSHLNYTCGAENSTGASQARPHAYYALSYCALILAIVFGNGLVCMAVLKERAL
QTTTNYLVVSLAVADLLVATLVMPWVVYLEVTGGVWNFSRICCDVFVTLDVMMCTASILN
LCAISIDRYTAVVMPVHYQHGTGQSSCRRVALMITAVWVLAFAVSCPLLFGFNTTGDPTV
CSISNPDFVIYSSVVSFYLPFGVTVLVYARIYVVLKQRRRKRILTRQNSQCNSVRPGFPQ
QTLSPDPAHLELKRYYSICQDTALGGPGFQERGGELKREEKTRNSLSPTIAPKLSLEVRK
LSNGRLSTSLKLGPLQPRGVPLREKKATQMVAIVLGAFIVCWLPFFLTHVLNTHCQTCHV
SPELYSATTWLGYVNSALNPVIYTTFNIEFRKAFLKILSC
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| BDBM50207049 |
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| n/a |
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| Name | BDBM50207049 |
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| Synonyms: | CHEMBL3919497 |
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| Type | Small organic molecule |
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| Emp. Form. | C20H22N2O3S |
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| Mol. Mass. | 370.465 |
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| SMILES | CN(C)[C@@H]1[C@@H](CCO)c2cc3ccn(c3cc12)S(=O)(=O)c1ccccc1 |r| |
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| Structure | 
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