| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Lysophosphatidic acid receptor 4 |
|---|
| Ligand | BDBM50233165 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | ChEMBL_1649816 (CHEMBL3998950) |
|---|
| EC50 | 570±n/a nM |
|---|
| Citation |  Banerjee, S; Norman, DD; Lee, SC; Parrill, AL; Pham, TC; Baker, DL; Tigyi, GJ; Miller, DD Highly Potent Non-Carboxylic Acid Autotaxin Inhibitors Reduce Melanoma Metastasis and Chemotherapeutic Resistance of Breast Cancer Stem Cells. J Med Chem60:1309-1324 (2017) [PubMed] Article |
|---|
| More Info.: | Get all data from this article, Assay Method |
|---|
| |
| Lysophosphatidic acid receptor 4 |
|---|
| Name: | Lysophosphatidic acid receptor 4 |
|---|
| Synonyms: | GPR23 | LPA4 | LPAR4 | LPAR4_HUMAN | P2RY9 |
|---|
| Type: | PROTEIN |
|---|
| Mol. Mass.: | 41910.31 |
|---|
| Organism: | Homo sapiens (Human) |
|---|
| Description: | ChEMBL_946257 |
|---|
| Residue: | 370 |
|---|
| Sequence: | MGDRRFIDFQFQDSNSSLRPRLGNATANNTCIVDDSFKYNLNGAVYSVVFILGLITNSVS
LFVFCFRMKMRSETAIFITNLAVSDLLFVCTLPFKIFYNFNRHWPFGDTLCKISGTAFLT
NIYGSMLFLTCISVDRFLAIVYPFRSRTIRTRRNSAIVCAGVWILVLSGGISASLFSTTN
VNNATTTCFEGFSKRVWKTYLSKITIFIEVVGFIIPLILNVSCSSVVLRTLRKPATLSQI
GTNKKKVLKMITVHMAVFVVCFVPYNSVLFLYALVRSQAITNCFLERFAKIMYPITLCLA
TLNCCFDPFIYYFTLESFQKSFYINAHIRMESLFKTETPLTTKPSLPAIQEEVSDQTTNN
GGELMLESTF
|
|
|
|---|
| BDBM50233165 |
|---|
| n/a |
|---|
| Name | BDBM50233165 |
|---|
| Synonyms: | CHEMBL1222042 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C21H41O7P |
|---|
| Mol. Mass. | 436.5198 |
|---|
| SMILES | CCCCCCCC\C=C/CCCCCCCC(=O)OCC(O)COP(O)(O)=O |
|---|
| Structure | 
|
|---|
Search and Browse
