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TargetMu-type opioid receptor
LigandBDBM50236872
Substrate/Competitorn/a
Meas. Tech.ChEBML_1659530
Ki 1230±n/a nM
Citation Soeberdt, MMolenveld, PStorcken, RPBouzanne des Mazery, RSterk, GJAutar, RBolster, MGWagner, CAerts, SNvan Holst, FRWegert, ATangherlini, GFrehland, BSchepmann, DMetze, DLotts, TKnie, ULin, KYHuang, TYLai, CCStänder, SWünsch, BAbels, C Design and Synthesis of Enantiomerically Pure Decahydroquinoxalines as Potent and Selective¿-Opioid Receptor Agonists with Anti-Inflammatory Activity in Vivo. J Med Chem60:2526-2551 (2017) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Mu-type opioid receptor
Name:Mu-type opioid receptor
Synonyms:M-OR-1 | MOR-1 | Mu opioid receptor | Mu-type opioid receptor (Mu) | OPIATE Mu | OPRM1 | OPRM_CAVPO
Type:Enzyme Catalytic Domain
Mol. Mass.:11165.58
Organism:GUINEA PIG
Description:P97266
Residue:98
Sequence:
YTKMKTATNIYIFNLALADALATSTLPFQSVNYLMGTWPFGTILCKIVISIDYYNMFTSI
FTLCTMSVDRYIAVCHPVKALDFRTPRNAKTVNVCNWI
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  Blast E-value cutoff:
BDBM50236872
n/a
NameBDBM50236872
Synonyms:CHEMBL4072972
TypeSmall organic molecule
Emp. Form.C23H31Cl2N3O3
Mol. Mass.468.417
SMILES[H][C@]12CCC[C@H](N3CCCC3)[C@@]1([H])N(CCN2CC(=O)OC)C(=O)Cc1ccc(Cl)c(Cl)c1 |r|
Structure
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