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TargetMu-type opioid receptor
LigandBDBM50236886
Substrate/Competitorn/a
Meas. Tech.ChEMBL_1659530
Ki 830±n/a nM
Citation Soeberdt MMolenveld PStorcken RPBouzanne des Mazery RSterk GJAutar RBolster MGWagner CAerts SNvan Holst FRWegert ATangherlini GFrehland BSchepmann DMetze DLotts TKnie ULin KYHuang TYLai CCStänder SWünsch BAbels C Design and Synthesis of Enantiomerically Pure Decahydroquinoxalines as Potent and Selective¿-Opioid Receptor Agonists with Anti-Inflammatory Activity in Vivo. J Med Chem 60:2526-2551 (2017) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Mu-type opioid receptor
Name:Mu-type opioid receptor
Synonyms:M-OR-1 | MOR-1 | Mu opioid receptor | Mu-type opioid receptor (Mu) | OPIATE Mu | OPRM1
Type:Enzyme Catalytic Domain
Mol. Mass.:11165.58
Organism:GUINEA PIG
Description:P97266
Residue:98
Sequence:
YTKMKTATNIYIFNLALADALATSTLPFQSVNYLMGTWPFGTILCKIVISIDYYNMFTSI
FTLCTMSVDRYIAVCHPVKALDFRTPRNAKTVNVCNWI
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  Blast E-value cutoff:
BDBM50236886
n/a
NameBDBM50236886
Synonyms:CHEMBL4099849
TypeSmall organic molecule
Emp. Form.C24H33Cl2N3O3
Mol. Mass.482.443
SMILES[H][C@]12CCC[C@H](N3CCCC3)[C@@]1([H])N(CCN2CC(=O)OCC)C(=O)Cc1ccc(Cl)c(Cl)c1 |r|
Structure
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