Reaction Details |
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Target | 5-hydroxytryptamine receptor 5A |
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Ligand | BDBM81498 |
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Substrate/Competitor | n/a |
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Ki | 316.22±n/a nM |
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Comments | PDSP_1643 |
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Citation | Matthes, H; Boschert, U; Amlaiky, N; Grailhe, R; Plassat, JL; Muscatelli, F; Mattei, MG; Hen, R Mouse 5-hydroxytryptamine5A and 5-hydroxytryptamine5B receptors define a new family of serotonin receptors: cloning, functional expression, and chromosomal localization. Mol Pharmacol43:313-9 (1993) [PubMed] |
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More Info.: | Get all data from this article |
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5-hydroxytryptamine receptor 5A |
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Name: | 5-hydroxytryptamine receptor 5A |
Synonyms: | 5-HT-5 | 5-HT-5A | 5-HT5 | 5-HT5a | 5-hydroxytryptamine receptor 5A | 5HT5A_MOUSE | 5ht5a | Htr5a | Serotonin 5a (5-HT5a) receptor | Serotonin receptor 5A |
Type: | Enzyme Catalytic Domain |
Mol. Mass.: | 40749.33 |
Organism: | MOUSE |
Description: | 5-HT5 0 MOUSE::P30966 |
Residue: | 357 |
Sequence: | MDLPVNLTSFSLSTPSSLEPNRSLDTEVLRPSRPFLSAFRVLVLTLLGFLAAATFTWNLL
VLATILKVRTFHRVPHNLVASMAISDVLVAVLVMPLSLVHELSGRRWQLGRRLCQLWIAC
DVLCCTASIWNVTAIALDRYWSITRHLEYTLRTRKRVSNVMILLTWALSTVISLAPLLFG
WGETYSEPSEECQVSREPSYTVFSTVGAFYLPLCVVLFVYWKIYRAAKFRMGSRKTNSVS
PVPEAVEVKNATQHPQMVFTVRHATVTFQTEGDTWREQKEQRAALMVGILIGVFVLCWFP
FFVTELISPLCSWDVPAIWKSIFLWLGYSNSFFNPLIYTAFNRSYSSAFKVFFSKQQ
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BDBM81498 |
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n/a |
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Name | BDBM81498 |
Synonyms: | 5-Methoxy-3-(1,2,3,6-tetrahydro-pyridin-4-yl)-1H-indole(RU-24969) | CAS_108028 | CHEMBL18785 | NSC_108028 | RU 24969 |
Type | Small organic molecule |
Emp. Form. | C14H16N2O |
Mol. Mass. | 228.2896 |
SMILES | COc1ccc2[nH]cc(C3=CCNCC3)c2c1 |t:9| |
Structure |
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