| Reaction Details |
|---|
 | Report a problem with these data |
| Target | 5-hydroxytryptamine receptor 2A |
|---|
| Ligand | BDBM84930 |
|---|
| Substrate/Competitor | n/a |
|---|
| Ki | 33.1±n/a nM |
|---|
| Comments | PDSP_1151 |
|---|
| Citation |  Nelson, DL; Lucaites, VL; Audia, JE; Nissen, JS; Wainscott, DB Species differences in the pharmacology of the 5-hydroxytryptamine2 receptor: structurally specific differentiation by ergolines and tryptamines. J Pharmacol Exp Ther265:1272-9 (1993) [PubMed] |
|---|
| More Info.: | Get all data from this article |
|---|
| |
| 5-hydroxytryptamine receptor 2A |
|---|
| Name: | 5-hydroxytryptamine receptor 2A |
|---|
| Synonyms: | 5-HT2 | 5HT2A_MACMU | HTR2A |
|---|
| Type: | Enzyme Catalytic Domain |
|---|
| Mol. Mass.: | 52607.65 |
|---|
| Organism: | Monkey |
|---|
| Description: | 5-HT2 0 Monkey::P50128 |
|---|
| Residue: | 471 |
|---|
| Sequence: | MDILCEENTSLSSTTNSLMQLNEDTRLYSNDFNSGEANTSDAFNWTVESENRTNLSCEGC
LSPSCLSLLHLQEKNWSALLTAVVIILTIAGNILVIMAVSLEKKLQNATNYFLMSLAIAD
MLLGFLVMPVSMLTILYGYRWPLPSKLCAVWIYLDVLFSTASIMHLCAISLDRYVAIQNP
IHHSRFNSRTKAFLKIIAVWTISVGISMPIPVFGLQDDSKVFKEGSCLLADDNFVLIGSF
VSFFIPLTIMVITYFLTIKSLQKEATLCVSDLGTRAKLASFSFLPQSSLSSEKLFQRSIH
RDPGSYTGRRTMQSISNEQKACKVLGIVFFLFVVMWCPFFITNIMAVICKESCNEDVIGA
LLNVFVWIGYLSSAVNPLVYTLFNKTYRSAFSRYIQCQYKENKKPLQLILVNTIPALAYK
SSQLQMGQKKNSKQDAKTTDNDCSMVALGKQHSEDASKDNSDGVNEKVSCV
|
|
|
|---|
| BDBM84930 |
|---|
| n/a |
|---|
| Name | BDBM84930 |
|---|
| Synonyms: | CAS_60634-51-7 | LY 53857 | NSC_107989 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C23H32N2O3 |
|---|
| Mol. Mass. | 384.5118 |
|---|
| SMILES | CC(O)C(C)OC(=O)C1CC2C(Cc3cn(C(C)C)c4cccc2c34)N(C)C1 |
|---|
| Structure | 
|
|---|
Search and Browse
