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| Reaction Details | |||
|---|---|---|---|
 | Report a problem with these data | ||
| Target | 5-hydroxytryptamine receptor 5A | ||
| Ligand | BDBM50031942 | ||
| Substrate/Competitor | n/a | ||
| Ki | 500±n/a nM | ||
| Comments | PDSP_1230 | ||
| Citation |  Weiss, HM; Haase, W; Michel, H; Reiländer, H Expression of functional mouse 5-HT5A serotonin receptor in the methylotrophic yeast Pichia pastoris: pharmacological characterization and localization. FEBS Lett377:451-6 (1995) [PubMed] Article | ||
| More Info.: | Get all data from this article | ||
| 5-hydroxytryptamine receptor 5A | |||
| Name: | 5-hydroxytryptamine receptor 5A | ||
| Synonyms: | 5-HT-5 | 5-HT-5A | 5-HT5 | 5-HT5a | 5-hydroxytryptamine receptor 5A | 5HT5A_MOUSE | 5ht5a | Htr5a | Serotonin 5a (5-HT5a) receptor | Serotonin receptor 5A | ||
| Type: | Enzyme Catalytic Domain | ||
| Mol. Mass.: | 40749.33 | ||
| Organism: | MOUSE | ||
| Description: | 5-HT5 0 MOUSE::P30966 | ||
| Residue: | 357 | ||
| Sequence: |
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| BDBM50031942 | |||
| n/a | |||
| Name | BDBM50031942 | ||
| Synonyms: | (6aR,9R)-4,6a,7-Trimethyl-4,6,6a,7,8,9-hexahydro-indolo[4,3-fg]quinoline-9-carboxylic acid (1-hydroxymethyl-propyl)-amide | (6aR,9R)-4,7-Dimethyl-4,6,6a,7,8,9-hexahydro-indolo[4,3-fg]quinoline-9-carboxylic acid ((S)-1-hydroxymethyl-propyl)-amide | (6aR,9R)-4-Methyl-4,6,6a,7,8,9-hexahydro-indolo[4,3-fg]quinoline-9-carboxylic acid (1-hydroxymethyl-propyl)-amide | (6aR,9R)-5,7-Dimethyl-4,6,6a,7,8,9-hexahydro-indolo[4,3-fg]quinoline-9-carboxylic acid diethylamide | (methylsergide)4,7-Dimethyl-4,6,6a,7,8,9-hexahydro-indolo[4,3-fg]quinoline-9-carboxylic acid (1-hydroxymethyl-propyl)-amide | 4,7-Dimethyl-4,6,6a,7,8,9-hexahydro-indolo[4,3-fg]quinoline-9-carboxylic acid (1-hydroxymethyl-propyl)-amide | CHEMBL1065 | METHYSERGIDE | Sansert | ||
| Type | Small organic molecule | ||
| Emp. Form. | C21H27N3O2 | ||
| Mol. Mass. | 353.458 | ||
| SMILES | CC[C@@H](CO)NC(=O)[C@H]1CN(C)[C@@H]2Cc3cn(C)c4cccc(C2=C1)c34 |r,c:24| | ||
| Structure | 
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