Reaction Details |
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Target | Neuropeptide Y receptor type 5 |
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Ligand | BDBM50015490 |
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Substrate/Competitor | n/a |
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Ki | 4.3±n/a nM |
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Comments | PDSP_1370 |
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Citation | Weinberg, DH; Sirinathsinghji, DJ; Tan, CP; Shiao, LL; Morin, N; Rigby, MR; Heavens, RH; Rapoport, DR; Bayne, ML; Cascieri, MA; Strader, CD; Linemeyer, DL; MacNeil, DJ Cloning and expression of a novel neuropeptide Y receptor. J Biol Chem271:16435-8 (1996) [PubMed] Article |
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More Info.: | Get all data from this article |
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Neuropeptide Y receptor type 5 |
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Name: | Neuropeptide Y receptor type 5 |
Synonyms: | NPY-Y5 | NPY5R_MOUSE | Neuropeptide Y receptor Y5 | Neuropeptide Y receptor type 5 (NPY Y5) | Npy5 | Npy5r |
Type: | Enzyme |
Mol. Mass.: | 52807.91 |
Organism: | Mus musculus (Mouse) |
Description: | O70342 |
Residue: | 466 |
Sequence: | MEVKLEEHFNKTFVTENNTAASQNTASPAWEDYRGTENNTSAARNTAFPVWEDYRGSVDD
LQYFLIGLYTFVSLLGFMGNLLILMAVMKKRNQKTTVNFLIGNLAFSDILVVLFCSPFTL
TSVLLDQWMFGKAMCHIMPFLQCVSVLVSTLILISIAIVRYHMIKHPISNNLTANHGYFL
IATVWTLGFAICSPLPVFHSLVELKETFGSALLSSKYLCVESWPSDSYRIAFTISLLLVQ
YILPLVCLTVSHTSVCRSISCGLSHKENRLEENEMINLTLHPSKKSRDQAKPPSTQKWSY
SFIRKHRRRYSKKTACVLPAPAGPSQEKHLTVPENPGSVRSQLSPSSKVIPGVPICFEVK
PEESSDAQEMRVKRSLTRIKKRSRSVFYRLTILILVFAVSWMPLHVFHVVTDFNDNLISN
RHFKLVYCICHLLGMMSCCLNPILYGFLNNGIKADLRALIHCLHMS
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BDBM50015490 |
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n/a |
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Name | BDBM50015490 |
Synonyms: | CHEMBL438945 | H-YPSKPDNPGEDAPAEDMARYYSALRHYINLITRQRY-NH2 | NPY | NPY, human | NPY, human, rat | Tyr-Pro-Ser-Lys-Pro-Asp-Asn-Pro-Gly-Glu-Asp-Ala-Pro- Ala-Glu-Asp-Met-Ala-Arg-Tyr-Tyr-Ser-Ala-Leu-Arg-His- Tyr-Ile-Asn-Leu-Ile-Thr-Arg-Gln-Arg-Tyr-NH2 (NPY) | human Neuropeptide Y |
Type | Small organic molecule |
Emp. Form. | C189H285N55O57S |
Mol. Mass. | 4271.685 |
SMILES | n/a |
Structure |
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