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TargetGamma-aminobutyric acid receptor subunit alpha-6
LigandBDBM50244035
Substrate/Competitorn/a
Ki 4461.28±n/a nM
CommentsPDSP_350
Citation Yang, WDrewe, JALan, NC Cloning and characterization of the human GABAA receptor alpha 4 subunit: identification of a unique diazepam-insensitive binding site. Eur J Pharmacol291:319-25 (1995) [PubMed]  Article
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Gamma-aminobutyric acid receptor subunit alpha-6
Name:Gamma-aminobutyric acid receptor subunit alpha-6
Synonyms:GABA A alpha6 | GABA receptor alpha-6 subunit | GABRA6 | GBRA6_HUMAN
Type:Enzyme Catalytic Domain
Mol. Mass.:51029.60
Organism:Homo sapiens (Human)
Description:GABA A alpha6 0 HUMAN::Q16445
Residue:453
Sequence:
MASSLPWLCIILWLENALGKLEVEGNFYSENVSRILDNLLEGYDNRLRPGFGGAVTEVKT
DIYVTSFGPVSDVEMEYTMDVFFRQTWTDERLKFGGPTEILSLNNLMVSKIWTPDTFFRN
GKKSIAHNMTTPNKLFRIMQNGTILYTMRLTINADCPMRLVNFPMDGHACPLKFGSYAYP
KSEIIYTWKKGPLYSVEVPEESSSLLQYDLIGQTVSSETIKSNTGEYVIMTVYFHLQRKM
GYFMIQIYTPCIMTVILSQVSFWINKESVPARTVFGITTVLTMTTLSISARHSLPKVSYA
TAMDWFIAVCFAFVFSALIEFAAVNYFTNLQTQKAKRKAQFAAPPTVTISKATEPLEAEI
VLHPDSKYHLKKRITSLSLPIVSSSEANKVLTRAPILQSTPVTPPPLSPAFGGTSKIDQY
SRILFPVAFAGFNLVYWVVYLSKDTMEVSSSVE
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  Blast E-value cutoff:
BDBM50244035
n/a
NameBDBM50244035
Synonyms:Beta CCE | CHEMBL454606 | cid_105078 | ethyl 9H-pyrido[3,4-b]indole-3-carboxylate
TypeSmall organic molecule
Emp. Form.C14H12N2O2
Mol. Mass.240.2573
SMILESCCOC(=O)c1cc2c(cn1)[nH]c1ccccc21
Structure
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