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TargetGABA A receptor alpha-6/beta-2/gamma-2
LigandBDBM81951
Substrate/Competitorn/a
Ki 152.89±n/a nM
CommentsPDSP_689
Citation Yang WDrewe JALan NC Cloning and characterization of the human GABAA receptor alpha 4 subunit: identification of a unique diazepam-insensitive binding site. Eur J Pharmacol 291:319-25 (1995) [PubMed]  Article
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GABA A receptor alpha-6/beta-2/gamma-2
Name:Gamma-aminobutyric acid receptor subunit alpha-6/beta-3
Synonyms:GABA A Alpha6Beta2Gamma2 | GABA A Alpha6Beta3Gamma2 | GABA A alpha6 | GABA receptor alpha-6 subunit | Gamma-aminobutyric acid receptor subunit alpha-6
Type:Enzyme Catalytic Domain
Mol. Mass.:51029.60
Organism:Homo sapiens (Human)
Description:GABA A alpha6 0 HUMAN::Q16445
Residue:453
Sequence:
MASSLPWLCIILWLENALGKLEVEGNFYSENVSRILDNLLEGYDNRLRPGFGGAVTEVKT
DIYVTSFGPVSDVEMEYTMDVFFRQTWTDERLKFGGPTEILSLNNLMVSKIWTPDTFFRN
GKKSIAHNMTTPNKLFRIMQNGTILYTMRLTINADCPMRLVNFPMDGHACPLKFGSYAYP
KSEIIYTWKKGPLYSVEVPEESSSLLQYDLIGQTVSSETIKSNTGEYVIMTVYFHLQRKM
GYFMIQIYTPCIMTVILSQVSFWINKESVPARTVFGITTVLTMTTLSISARHSLPKVSYA
TAMDWFIAVCFAFVFSALIEFAAVNYFTNLQTQKAKRKAQFAAPPTVTISKATEPLEAEI
VLHPDSKYHLKKRITSLSLPIVSSSEANKVLTRAPILQSTPVTPPPLSPAFGGTSKIDQY
SRILFPVAFAGFNLVYWVVYLSKDTMEVSSSVE
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BDBM81951
n/a
NameBDBM81951
Synonyms:CAS_104999 | DMCM | NSC_104999
TypeSmall organic molecule
Emp. Form.C17H18N2O4
Mol. Mass.314.3358
SMILESCCc1c(ncc2[nH]c3cc(OC)c(OC)cc3c12)C(=O)OC
Structure
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