Ki Summary BindingDB logo
myBDB logout
Reaction Details
Report a problem with these data
TargetGamma-aminobutyric acid receptor subunit alpha-6
LigandBDBM84955
Substrate/Competitorn/a
Ki 2506.73±n/a nM
CommentsPDSP_820
Citation Yang, WDrewe, JALan, NC Cloning and characterization of the human GABAA receptor alpha 4 subunit: identification of a unique diazepam-insensitive binding site. Eur J Pharmacol291:319-25 (1995) [PubMed]  Article
More Info.:Get all data from this article
 
Gamma-aminobutyric acid receptor subunit alpha-6
Name:Gamma-aminobutyric acid receptor subunit alpha-6
Synonyms:GABA A alpha6 | GABA receptor alpha-6 subunit | GABRA6 | GBRA6_HUMAN
Type:Enzyme Catalytic Domain
Mol. Mass.:51029.60
Organism:Homo sapiens (Human)
Description:GABA A alpha6 0 HUMAN::Q16445
Residue:453
Sequence:
MASSLPWLCIILWLENALGKLEVEGNFYSENVSRILDNLLEGYDNRLRPGFGGAVTEVKT
DIYVTSFGPVSDVEMEYTMDVFFRQTWTDERLKFGGPTEILSLNNLMVSKIWTPDTFFRN
GKKSIAHNMTTPNKLFRIMQNGTILYTMRLTINADCPMRLVNFPMDGHACPLKFGSYAYP
KSEIIYTWKKGPLYSVEVPEESSSLLQYDLIGQTVSSETIKSNTGEYVIMTVYFHLQRKM
GYFMIQIYTPCIMTVILSQVSFWINKESVPARTVFGITTVLTMTTLSISARHSLPKVSYA
TAMDWFIAVCFAFVFSALIEFAAVNYFTNLQTQKAKRKAQFAAPPTVTISKATEPLEAEI
VLHPDSKYHLKKRITSLSLPIVSSSEANKVLTRAPILQSTPVTPPPLSPAFGGTSKIDQY
SRILFPVAFAGFNLVYWVVYLSKDTMEVSSSVE
Blast this sequence in BindingDB or PDB
  Blast E-value cutoff:
BDBM84955
n/a
NameBDBM84955
Synonyms:CAS_4375 | FG 7142 | NSC_4375
TypeSmall organic molecule
Emp. Form.C13H11N3O
Mol. Mass.225.2459
SMILESCNC(=O)c1cc2c(cn1)[nH]c1ccccc21
Structure
Search PDB for entries with ligand similarity:Similarity to this molecule at least: