| Reaction Details |
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 | Report a problem with these data |
| Target | Histamine H2 receptor |
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| Ligand | BDBM82472 |
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| Substrate/Competitor | n/a |
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| Ki | >10000±n/a nM |
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| Comments | PDSP_456 |
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| Citation |  Kennett, GA; Bright, F; Trail, B; Baxter, GS; Blackburn, TP Effects of the 5-HT2B receptor agonist, BW 723C86, on three rat models of anxiety. Br J Pharmacol117:1443-8 (1996) [PubMed] Article |
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| More Info.: | Get all data from this article |
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| Histamine H2 receptor |
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| Name: | Histamine H2 receptor |
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| Synonyms: | HISTAMINE H2 | HRH2_MOUSE | Hrh2 | Hrh2 protein |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 44816.27 |
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| Organism: | Mus musculus |
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| Description: | P97292 |
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| Residue: | 397 |
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| Sequence: | MEPNGTVHSCCLDSIALKVTISVVLTTLIFITVAGNVVVCLAVSLNRRLRSLTNCFIVSL
AATDLLLGLLVMPFSAIYQLSFKWSFGQVFCNIYTSLDVMLCTASILNLFMISLDRYCAV
TDPLRYPVLVTPVRVAISLVFIWVISITLSFLSIHLGWNSRNGTRGGNDTFKCKVQVNEV
YGLVDGMVTFYLPLLIMCVTYYRIFKIAREQAKRINHISSWKAATIREHKATVTLAAVMG
AFIVCWFPYFTAFVYRGLRGDDAVNEVVEGIVLWLGYANSALNPILYATLNRDFRMAYQQ
LFHCKLASHNSHKTSLRLNNSLLSRSQSREGRWQEEKPLKLQVWSGTELTHPQGSPVRTR
LSHSSCLLSLSLLSFIWKLGTWIHHRRPFQPSLHISA
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| BDBM82472 |
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| n/a |
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| Name | BDBM82472 |
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| Synonyms: | BW-723C86 | CAS_5311036 | NSC_5311036 |
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| Type | Small organic molecule |
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| Emp. Form. | C16H18N2OS |
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| Mol. Mass. | 286.392 |
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| SMILES | CC(N)Cc1c[nH]c2ccc(OCc3cccs3)cc12 |
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| Structure | 
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