| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Histamine H2 receptor |
|---|
| Ligand | BDBM82472 |
|---|
| Substrate/Competitor | n/a |
|---|
| Ki | >10000±n/a nM |
|---|
| Comments | PDSP_456 |
|---|
| Citation |  Baxter, GS Novel discriminatory ligands for 5-HT2B receptors. Behav Brain Res73:149-52 (1996) [PubMed] Article |
|---|
| More Info.: | Get all data from this article |
|---|
| |
| Histamine H2 receptor |
|---|
| Name: | Histamine H2 receptor |
|---|
| Synonyms: | HISTAMINE H2 | HRH2 |
|---|
| Type: | Enzyme Catalytic Domain |
|---|
| Mol. Mass.: | 40972.37 |
|---|
| Organism: | RABBIT |
|---|
| Description: | HISTAMINE H2 HRH2 RABBIT::G1TWL8 |
|---|
| Residue: | 367 |
|---|
| Sequence: | MEPNDTANDTASSSCLESTAFKVTLSVVLTILILITAAGNVVVCLAVGLNRRLRSLTNCF
IVSLAITDLLLGLLVLPFSAIYQLSCRWSFGKVFCNIYISLDVMLCTASILNLFMISIDR
YCAVTDPLRYPVLVTPGRVTISLVSIWVISITLSFLSIHLGWNSRNTTSEGHHTSPKCKF
QVNEVYGLVDGLVTFYLPLLIMCVTYYRIFKIAREQARRINHISSWQAATIREHKATVTL
AAVMGAFIVCWFPYFTTFVYRGLKGDDAINEVVEAVVLWLGYANSALNPILYAALNRDFR
NAYQQLFCCRLAGRGSHETCLRFNNALLPKSQSQEPRRQEEKPLKLQVWSGTEATAPQGA
TDRVFGE
|
|
|
|---|
| BDBM82472 |
|---|
| n/a |
|---|
| Name | BDBM82472 |
|---|
| Synonyms: | BW-723C86 | CAS_5311036 | NSC_5311036 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C16H18N2OS |
|---|
| Mol. Mass. | 286.392 |
|---|
| SMILES | CC(N)Cc1c[nH]c2ccc(OCc3cccs3)cc12 |
|---|
| Structure | 
|
|---|
Search and Browse
