| Reaction Details |
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 | Report a problem with these data |
| Target | Beta-arrestin-1 |
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| Ligand | BDBM81483 |
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| Substrate/Competitor | n/a |
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| Ki | 1000±n/a nM |
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| Comments | PDSP_1499 |
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| Citation |  Schotte, A; Janssen, PF; Gommeren, W; Luyten, WH; Van Gompel, P; Lesage, AS; De Loore, K; Leysen, JE Risperidone compared with new and reference antipsychotic drugs: in vitro and in vivo receptor binding. Psychopharmacology (Berl)124:57-73 (1996) [PubMed] Article |
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| More Info.: | Get all data from this article |
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| Beta-arrestin-1 |
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| Name: | Beta-arrestin-1 |
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| Synonyms: | ARRB1 | ARRB1_RABIT | Beta-arrestin-1 | Cholinergic, muscarinic | OPIATE Delta | PAF Platelet activating factor |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 46360.54 |
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| Organism: | RABBIT |
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| Description: | Cholinergic, muscarinic 0 RABBIT::Q95223 |
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| Residue: | 410 |
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| Sequence: | MGDKGTRVFKKASPNGKLTVYLGKRGFVDHIDLVDPVDGVVLVDPEYLKERRVYVTLTCA
FRYGREDLDVLGLTFRKDLFVANVQSFPPAPEDKKPLTRLQERLIKKLGEHAYPFTFEIP
PKLPCSVTLQPGPEDTGKACGVDYEVKAFCAENLEEKIHKRNSVRLVIRKVQYAPERPGP
HPTAETTRLFLMSDKPLHLEASLDKEIYYHGEPIIVNVHVTNNTNKTVKKIKISVRQYAD
ICLFNTAQYKCPVAMEEADDTVAPSSTFCKVYTLTPFLANNREKRGLALDGKLKHEDTNL
ASSTLMREGANREILGIIVSYKVKVKLVVSRGGDVAVELPFTLMHPKPKEEPPHREVPEN
ETPVDTNLIELDTNDDDIVFEDFARQRLKGMKDDKEEEDDVTGSPRLNDR
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| BDBM81483 |
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| n/a |
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| Name | BDBM81483 |
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| Synonyms: | CAS_1893-33-0 | NSC_4830 | PIPAMPERONE |
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| Type | Small organic molecule |
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| Emp. Form. | C21H30FN3O2 |
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| Mol. Mass. | 375.4802 |
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| SMILES | NC(=O)C1(CCN(CCCC(=O)c2ccc(F)cc2)CC1)N1CCCCC1 |
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| Structure | 
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