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TargetHTR4
LigandBDBM29525
Substrate/Competitorn/a
Ki 0.31±n/a nM
CommentsPDSP_880
Citation Claeysen SSebben MJournot LBockaert JDumuis A Cloning, expression and pharmacology of the mouse 5-HT(4L) receptor. FEBS Lett 398:19-25 (1996) [PubMed]  Article
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HTR4
Name:HTR4
Synonyms:5-HT-4 | 5-HT4 | 5-HT4L | 5-hydroxytryptamine receptor 4 | Serotonin 4 (5-HT4) receptor | Serotonin receptor 4
Type:Enzyme Catalytic Domain
Mol. Mass.:43970.99
Organism:MOUSE
Description:5-HT4 HTR4 MOUSE::P97288
Residue:388
Sequence:
MDKLDANVSSNEGFRSVEKVVLLTFLAVVILMAILGNLLVMVAVCRDRQLRKIKTNYFIV
SLAFADLLVSVLVMPFGAIELVQDIWAYGEMFCLVRTSLDVLLTTASIFHLCCISLDRYY
AICCQPLVYRNKMTPLRIALMLGGCWVLPMFISFLPIMQGWNNIGIVDVIEKRKFSHNSN
STWCVFMVNKPYAITCSVVAFYIPFLLMVLAYYRIYVTAKEHAQQIQMLQRAGATSESRP
QPADQHSTHRMRTETKAAKTLCVIMGCFCFCWAPFFVTNIVDPFIDYTVPEQVWTAFLWL
GYINSGLNPFLYAFLNKSFRRAFLIILCCDDERYKRPPILGQTVPCSTTTINGSTHVLRD
TVECGGQWESRCHLTATSPLVAAQPSDT
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BDBM29525
n/a
NameBDBM29525
Synonyms:3H-GR113808 | CHEMBL518682 | GR 113808 | [3H] GR 113808 | [3H]GR113808
Typeradiolabeled ligand
Emp. Form.C19H27N3O4S
Mol. Mass.393.5
SMILESCn1cc(C(=O)OCC2CCN(CCNS(C)(=O)=O)CC2)c2ccccc12
Structure
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