| Reaction Details |
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 | Report a problem with these data |
| Target | Adenosine receptor A3 |
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| Ligand | BDBM21173 |
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| Substrate/Competitor | n/a |
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| Ki | 1120±n/a nM |
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| Comments | PDSP_739 |
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| Citation |  Hill, RJ; Oleynek, JJ; Hoth, CF; Kiron, MA; Weng, W; Wester, RT; Tracey, WR; Knight, DR; Buchholz, RA; Kennedy, SP Cloning, expression and pharmacological characterization of rabbit adenosine A1 and A3 receptors. J Pharmacol Exp Ther280:122-8 (1997) [PubMed] |
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| More Info.: | Get all data from this article |
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| Adenosine receptor A3 |
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| Name: | Adenosine receptor A3 |
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| Synonyms: | AA3R_RABIT | ADENOSINE A3 | ADORA3 |
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| Type: | Protein |
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| Mol. Mass.: | 36319.35 |
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| Organism: | Oryctolagus cuniculus (rabbit) |
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| Description: | O02667 |
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| Residue: | 319 |
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| Sequence: | MPDNSTTLFLAIRASYIVFEIVIGVCAVVGNVLVIWVIKLNPSLKTTTFYFIFSLALADI
AVGFLVMPLAIVISLGITIGFYSCLVMSCLLLVFTHASIMSLLAIAVDRYLRVKLTVRYR
RVTTQRRIWLALGLCWVVSLLVGFTPMFGWNMKPTLESARNYSDFQCKFDSVIPMEYMVF
FSFFTWILIPLLLMCALYVYIFYIIRNKLVQSFSSFKETGAFYRREFKTAKSLFLVLALF
AGCWLPLSIINCVTYFKCKVPDVVLLVGILLSHANSMMNPIVYACKIQKFKETYLLIFKA
RVTCQPSDSLDPSSEQNSE
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| BDBM21173 |
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| n/a |
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| Name | BDBM21173 |
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| Synonyms: | 1,3-dipropyl-8-cyclopentylxanthine | 8-cyclopentyl-1,3-dipropyl-2,3,6,7-tetrahydro-1H-purine-2,6-dione | CHEMBL183 | DPCPX | PD116948 | [3H]DPCPX |
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| Type | radiolabeled ligand |
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| Emp. Form. | C16H24N4O2 |
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| Mol. Mass. | 304.3874 |
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| SMILES | CCCn1c2nc([nH]c2c(=O)n(CCC)c1=O)C1CCCC1 |
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| Structure | 
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