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TargetMelatonin receptor
LigandBDBM85062
Substrate/Competitorn/a
Ki 15.8±n/a nM
CommentsPDSP_1261
Citation Dubocovich, MLMasana, MIIacob, SSauri, DM Melatonin receptor antagonists that differentiate between the human Mel1a and Mel1b recombinant subtypes are used to assess the pharmacological profile of the rabbit retina ML1 presynaptic heteroreceptor. Naunyn Schmiedebergs Arch Pharmacol355:365-75 (1997) [PubMed]  Article
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Melatonin receptor
Name:Melatonin receptor
Synonyms:Melatonin | Melatonin receptor
Type:Enzyme Catalytic Domain
Mol. Mass.:13287.02
Organism:RABBIT
Description:Q9BE38
Residue:114
Sequence:
MIWMLTLVAVMPNLHTGTLQYDPRVYSCTFSQSVSSAYTIAVVVFHFIIPMLMSSCCYLR
IWILVLQVRRRVKPDNKPKLKPQDFRNFITMFVVFVLFAICWAPLNFIVLLGRS
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BDBM85062
n/a
NameBDBM85062
Synonyms:Luzindole,N-propanoyl | N 0889 | N-0889 | N-[2-(2-Benzyl-1H-indol-3-yl)ethyl]propionamide
TypeSmall organic molecule
Emp. Form.C20H22N2O
Mol. Mass.306.4015
SMILESCCC(=O)NCCc1c(Cc2ccccc2)[nH]c2ccccc12
Structure
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