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TargetGalanin receptor type 1
LigandBDBM85073
Substrate/Competitorn/a
Ki 1±n/a nM
CommentsPDSP_3166
Citation Howard, ADTan, CShiao, LLPalyha, OCMcKee, KKWeinberg, DHFeighner, SDCascieri, MASmith, RGVan Der Ploeg, LHSullivan, KA Molecular cloning and characterization of a new receptor for galanin. FEBS Lett405:285-90 (1997) [PubMed]  Article
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Galanin receptor type 1
Name:Galanin receptor type 1
Synonyms:GALR1_RAT | Galanin R1 | Galanin receptor type 1 | Galnr | Galnr1 | Galr1
Type:Enzyme Catalytic Domain
Mol. Mass.:38883.91
Organism:RAT
Description:Galanin R1 GALR1 RAT::Q62805
Residue:346
Sequence:
MELAPVNLSEGNGSDPEPPAEPRPLFGIGVENFITLVVFGLIFAMGVLGNSLVITVLARS
KPGKPRSTTNLFILNLSIADLAYLLFCIPFQATVYALPTWVLGAFICKFIHYFFTVSMLV
SIFTLAAMSVDRYVAIVHSRRSSSLRVSRNALLGVGFIWALSIAMASPVAYYQRLFHRDS
NQTFCWEHWPNQLHKKAYVVCTFVFGYLLPLLLICFCYAKVLNHLHKKLKNMSKKSEASK
KKTAQTVLVVVVVFGISWLPHHVIHLWAEFGAFPLTPASFFFRITAHCLAYSNSSVNPII
YAFLSENFRKAYKQVFKCRVCNESPHGDAKEKNRIDTPPSTNCTHV
Blast this sequence in BindingDB or PDB
  Blast E-value cutoff:
BDBM85073
n/a
NameBDBM85073
Synonyms:CAS_3043476 | Galantide (M15) | NSC_3043476
TypeSmall organic molecule
Emp. Form.C23H30N2O3
Mol. Mass.382.4959
SMILESCOc1ccccc1N(CCOc1ccc(C)cc1)C(=O)CN1CCCCC1
Structure
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