Reaction Details |
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Target | Galanin receptor type 1 |
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Ligand | BDBM85073 |
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Substrate/Competitor | n/a |
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Ki | 1±n/a nM |
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Comments | PDSP_3166 |
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Citation | Howard, AD; Tan, C; Shiao, LL; Palyha, OC; McKee, KK; Weinberg, DH; Feighner, SD; Cascieri, MA; Smith, RG; Van Der Ploeg, LH; Sullivan, KA Molecular cloning and characterization of a new receptor for galanin. FEBS Lett405:285-90 (1997) [PubMed] Article |
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More Info.: | Get all data from this article |
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Galanin receptor type 1 |
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Name: | Galanin receptor type 1 |
Synonyms: | GALR1_RAT | Galanin R1 | Galanin receptor type 1 | Galnr | Galnr1 | Galr1 |
Type: | Enzyme Catalytic Domain |
Mol. Mass.: | 38883.91 |
Organism: | RAT |
Description: | Galanin R1 GALR1 RAT::Q62805 |
Residue: | 346 |
Sequence: | MELAPVNLSEGNGSDPEPPAEPRPLFGIGVENFITLVVFGLIFAMGVLGNSLVITVLARS
KPGKPRSTTNLFILNLSIADLAYLLFCIPFQATVYALPTWVLGAFICKFIHYFFTVSMLV
SIFTLAAMSVDRYVAIVHSRRSSSLRVSRNALLGVGFIWALSIAMASPVAYYQRLFHRDS
NQTFCWEHWPNQLHKKAYVVCTFVFGYLLPLLLICFCYAKVLNHLHKKLKNMSKKSEASK
KKTAQTVLVVVVVFGISWLPHHVIHLWAEFGAFPLTPASFFFRITAHCLAYSNSSVNPII
YAFLSENFRKAYKQVFKCRVCNESPHGDAKEKNRIDTPPSTNCTHV
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BDBM85073 |
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n/a |
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Name | BDBM85073 |
Synonyms: | CAS_3043476 | Galantide (M15) | NSC_3043476 |
Type | Small organic molecule |
Emp. Form. | C23H30N2O3 |
Mol. Mass. | 382.4959 |
SMILES | COc1ccccc1N(CCOc1ccc(C)cc1)C(=O)CN1CCCCC1 |
Structure |
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