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TargetGALR1
LigandBDBM50307254
Substrate/Competitorn/a
Ki 0.9±n/a nM
CommentsPDSP_1162
Citation Howard ADTan CShiao LLPalyha OCMcKee KKWeinberg DHFeighner SDCascieri MASmith RGVan Der Ploeg LHSullivan KA Molecular cloning and characterization of a new receptor for galanin. FEBS Lett 405:285-90 (1997) [PubMed]  Article
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GALR1
Name:GALR1
Synonyms:Galanin R1 | Galanin receptor type 1
Type:Enzyme Catalytic Domain
Mol. Mass.:38883.91
Organism:RAT
Description:Galanin R1 GALR1 RAT::Q62805
Residue:346
Sequence:
MELAPVNLSEGNGSDPEPPAEPRPLFGIGVENFITLVVFGLIFAMGVLGNSLVITVLARS
KPGKPRSTTNLFILNLSIADLAYLLFCIPFQATVYALPTWVLGAFICKFIHYFFTVSMLV
SIFTLAAMSVDRYVAIVHSRRSSSLRVSRNALLGVGFIWALSIAMASPVAYYQRLFHRDS
NQTFCWEHWPNQLHKKAYVVCTFVFGYLLPLLLICFCYAKVLNHLHKKLKNMSKKSEASK
KKTAQTVLVVVVVFGISWLPHHVIHLWAEFGAFPLTPASFFFRITAHCLAYSNSSVNPII
YAFLSENFRKAYKQVFKCRVCNESPHGDAKEKNRIDTPPSTNCTHV
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  Blast E-value cutoff:
BDBM50307254
n/a
NameBDBM50307254
Synonyms:CHEMBL604990 | GWTLNSAGYLLGPPPALALA-CONH2 | M40
TypeSmall organic molecule
Emp. Form.C94H145N23O24
Mol. Mass.1981.2968
SMILESCC(C)C[C@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)CN)[C@@H](C)O)C(=O)NCC(=O)N1CCC[C@H]1C(=O)N1CCC[C@H]1C(=O)N1CCC[C@H]1C(=O)N[C@@H](C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C)C(N)=O |r|
Structure
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