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TargetHTR1D
LigandBDBM86708
Substrate/Competitorn/a
Ki 2450±n/a nM
CommentsPDSP_1954
Citation Mos JVan Hest AVan Drimmelen MHerremans AHOlivier B The putative 5-HT1A receptor antagonist DU125530 blocks the discriminative stimulus of the 5-HT1A receptor agonist flesinoxan in pigeons. Eur J Pharmacol 325:145-53 (1997) [PubMed]  Article
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HTR1D
Name:HTR1D
Synonyms:5-HT1D
Type:Enzyme Catalytic Domain
Mol. Mass.:41807.41
Organism:pigeon
Description:5-HT1D HTR1D pigeon::A0A1V4JDN9
Residue:375
Sequence:
MTQYNHSAELALQSSANKSLNFTEALDERTLLGLKISLSVLLSVITLATILANVFVVITI
FLTRKLHTPANYLIGSLAVTDLLVSVLVMPISIAYTVTHTWAFGQVLCDIWLSSDITCCT
ASILHLCVIALDRYWAITDALEYAKRRTAGRAALMIAVVWMISVSISVPPFFWRQVKAHE
EIAKCAVNTDQISYTIYSTCGAFYIPSVLLLILYGRIYVAARSRILKPPSLYGKRFTTAH
LITGSAGSSLCSINASLHEGHSHPGGSPIFINHVQIKLADSVLERKRISAARERKATKTL
GIILGAFIFCWLPFFVMSLVLPICQDACWFHPILLDFFTWLGYLNSLINPVIYTAFNEEF
KQAFQNLIRVKKRLP
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  Blast E-value cutoff:
BDBM86708
n/a
NameBDBM86708
Synonyms:CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHEMBL537403 | NSC_104911 | WAY 100,635
TypeSmall organic molecule
Emp. Form.C25H34N4O2
Mol. Mass.422.5631
SMILESCOc1ccccc1N1CCN(CCN(C(=O)C2CCCCC2)c2ccccn2)CC1
Structure
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