| Reaction Details |
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 | Report a problem with these data |
| Target | Alpha-1A adrenergic receptor |
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| Ligand | BDBM50019443 |
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| Substrate/Competitor | n/a |
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| Ki | 7585±n/a nM |
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| Comments | PDSP_1495 |
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| Citation |  Mos, J; Van Hest, A; Van Drimmelen, M; Herremans, AH; Olivier, B The putative 5-HT1A receptor antagonist DU125530 blocks the discriminative stimulus of the 5-HT1A receptor agonist flesinoxan in pigeons. Eur J Pharmacol325:145-53 (1997) [PubMed] Article |
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| More Info.: | Get all data from this article |
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| Alpha-1A adrenergic receptor |
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| Name: | Alpha-1A adrenergic receptor |
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| Synonyms: | adrenergic Alpha1 |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 50699.64 |
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| Organism: | pigeon |
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| Description: | adrenergic Alpha1 0 pigeon::A0A1V4KJJ8 |
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| Residue: | 464 |
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| Sequence: | MAFLPGNSSDCSNCTHSVGPVNISKAILLGVILGGLIVFGVLGNILVILSVACHRHLQSV
THYYIINLAVADLLLTSTVLPFSATMEILGYWAFGRIFCNIWAAVDVLCCTASIMSLCII
SIDRYIGVSYPLRYPSIVTEKRGLLALLCVWALSLVISIGPLFGWKEPAPEDETICQITE
EPGYVLFSALGSFYLPLTIILVMYCRVYVVAKRENKGLSSGLKTERSHSEQVTLRIHRKN
APGASGSASNPKSKHHFSVRLLKFSREKKAAKTLGIVVGCFVLCWLPFFVVMPLGSFFPA
VKPPDTLFKITFWLGYLNSCINPIIYPCSSQEFKKAFQNVLRVQCLPRKQAAKKQSPSFN
LNHPASPSTESSRGVVRIPVGSGETFYKISKSDGVCEWKIFSAVQSMPAKTAVSKDCTAA
KVKSKGFLQECCCAGTSGNRGHENCKVPTIKIHTISLSESGEDV
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| BDBM50019443 |
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| n/a |
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| Name | BDBM50019443 |
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| Synonyms: | 1-(1H-Indol-4-yloxy)-3-isopropylamino-propan-2-ol | 1-(1H-Indol-4-yloxy)-3-isopropylamino-propan-2-ol((-)-Pindolol) | 1-(1H-Indol-4-yloxy)-3-isopropylamino-propan-2-ol(pindolol) | 1-(1H-indol-4-yloxy)-3-(isopropylamino)propan-2-ol | LB-46 | PINDOLOL | PINDOLOL,(-) | PRINODOLOL | VISKAZIDE | VISKEN |
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| Type | Small organic molecule |
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| Emp. Form. | C14H20N2O2 |
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| Mol. Mass. | 248.3208 |
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| SMILES | CC(C)NCC(O)COc1cccc2[nH]ccc12 |
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| Structure | 
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