| Reaction Details |
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 | Report a problem with these data |
| Target | Galanin receptor type 1 |
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| Ligand | BDBM50273367 |
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| Substrate/Competitor | n/a |
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| Ki | 2±n/a nM |
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| Comments | PDSP_855 |
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| Citation |  Smith, KE; Forray, C; Walker, MW; Jones, KA; Tamm, JA; Bard, J; Branchek, TA; Linemeyer, DL; Gerald, C Expression cloning of a rat hypothalamic galanin receptor coupled to phosphoinositide turnover. J Biol Chem272:24612-6 (1997) [PubMed] Article |
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| More Info.: | Get all data from this article |
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| Galanin receptor type 1 |
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| Name: | Galanin receptor type 1 |
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| Synonyms: | GALR1_RAT | Galanin R1 | Galanin receptor type 1 | Galnr | Galnr1 | Galr1 |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 38883.91 |
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| Organism: | RAT |
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| Description: | Galanin R1 GALR1 RAT::Q62805 |
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| Residue: | 346 |
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| Sequence: | MELAPVNLSEGNGSDPEPPAEPRPLFGIGVENFITLVVFGLIFAMGVLGNSLVITVLARS
KPGKPRSTTNLFILNLSIADLAYLLFCIPFQATVYALPTWVLGAFICKFIHYFFTVSMLV
SIFTLAAMSVDRYVAIVHSRRSSSLRVSRNALLGVGFIWALSIAMASPVAYYQRLFHRDS
NQTFCWEHWPNQLHKKAYVVCTFVFGYLLPLLLICFCYAKVLNHLHKKLKNMSKKSEASK
KKTAQTVLVVVVVFGISWLPHHVIHLWAEFGAFPLTPASFFFRITAHCLAYSNSSVNPII
YAFLSENFRKAYKQVFKCRVCNESPHGDAKEKNRIDTPPSTNCTHV
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| BDBM50273367 |
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| n/a |
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| Name | BDBM50273367 |
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| Synonyms: | (2S,3S)-2-((S)-2-((S)-2-((S)-1-(2-((S)-2-((S)-2-((S)-2-(2-((S)-2-((S)-2-((S)-4-amino-2-((S)-2-((2S,3R)-2-((S)-2-(2-aminoacetamido)-3-(1H-indol-3-yl)propanamido)-3-hydroxybutanamido)-4-methylpentanamido)-4-oxobutanamido)-3-hydroxypropanamido)propanamido)acetamido)-3-(4-hydroxyphenyl)propanamido)-4-methylpentanamido)-4-methylpentanamido)acetyl)pyrrolidine-2-carboxamido)-3-(1H-imidazol-5-yl)propanamido)propanamido)-3-methylpentanoic acid | CHEMBL499980 | Galanin (1-16) | Galanin (1-16), porcine | Galanin (1-16), rat |
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| Type | Small organic molecule |
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| Emp. Form. | C78H116N20O21 |
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| Mol. Mass. | 1669.877 |
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| SMILES | CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@@H]1CCCN1C(=O)CNC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)CN)[C@@H](C)O)C(O)=O |r| |
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| Structure | 
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