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TargetProstaglandin E2 receptor EP4 subtype
LigandBDBM85185
Substrate/Competitorn/a
Ki 43±n/a nM
CommentsPDSP_1463
Citation Kiriyama, MUshikubi, FKobayashi, THirata, MSugimoto, YNarumiya, S Ligand binding specificities of the eight types and subtypes of the mouse prostanoid receptors expressed in Chinese hamster ovary cells. Br J Pharmacol122:217-24 (1997) [PubMed]  Article
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Prostaglandin E2 receptor EP4 subtype
Name:Prostaglandin E2 receptor EP4 subtype
Synonyms:PE2R4_MOUSE | PGE receptor, EP4 subtype | Prostanoid EP4 receptor | Ptger4 | Ptgerep4
Type:G-protein coupled receptor
Mol. Mass.:56175.66
Organism:Mus musculus (Mouse)
Description:n/a
Residue:513
Sequence:
MAEVGGTIPRSNRELQRCVLLTTTIMSIPGVNASFSSTPERLNSPVTIPAVMFIFGVVGN
LVAIVVLCKSRKEQKETTFYTLVCGLAVTDLLGTLLVSPVTIATYMKGQWPGDQALCDYS
TFILLFFGLSGLSIICAMSIERYLAINHAYFYSHYVDKRLAGLTLFAIYASNVLFCALPN
MGLGRSERQYPGTWCFIDWTTNVTAYAAFSYMYAGFSSFLILATVLCNVLVCGALLRMHR
QFMRRTSLGTEQHHAAAAAAVASVACRGHAGASPALQRLSDFRRRRSFRRIAGAEIQMVI
LLIATSLVVLICSIPLVVRVFINQLYQPNVVKDISRNPDLQAIRIASVNPILDPWIYILL
RKTVLSKAIEKIKCLFCRIGGSGRDSSAQHCSESRRTSSAMSGHSRSFLARELKEISSTS
QTLLYLPDLTESSLGGRNLLPGSHGMGLTQADTTSLRTLRISETSDSSQGQDSESVLLVD
EVSGSHREEPASKGNSLQVTFPSETLKLSEKCI
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  Blast E-value cutoff:
BDBM85185
n/a
NameBDBM85185
Synonyms:PGE2,16,16-DIMETHYL
TypeSmall organic molecule
Emp. Form.C22H36O5
Mol. Mass.380.5182
SMILESCCCCC(C)(C)C(O)C=CC1C(O)CC(=O)C1CC=CCCCC(O)=O |w:9.8,19.19|
Structure
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