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TargetProstacyclin receptor
LigandBDBM85181
Substrate/Competitorn/a
Ki 16±n/a nM
CommentsPDSP_348
Citation Kiriyama, MUshikubi, FKobayashi, THirata, MSugimoto, YNarumiya, S Ligand binding specificities of the eight types and subtypes of the mouse prostanoid receptors expressed in Chinese hamster ovary cells. Br J Pharmacol122:217-24 (1997) [PubMed]  Article
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Prostacyclin receptor
Name:Prostacyclin receptor
Synonyms:PI2R_MOUSE | Prostacyclin receptor | Prostaglandin I | Prostaglandin I2 | Ptgir
Type:Enzyme Catalytic Domain
Mol. Mass.:44475.65
Organism:MOUSE
Description:Prostaglandin I2 PTGIR MOUSE::P43252
Residue:415
Sequence:
MMASDGHPGPPSVTPGSPLSAGGREWQGMAGSCWNITYVQDSVGPATSTLMFVAGVVGNG
LALGILGARRRSHPSAFAVLVTGLAVTDLLGTCFLSPAVFVAYARNSSLLGLAHGGTMLC
DTFAFAMTFFGLASTLILFAMAVERCLALSHPYLYAQLDGPRCARFALPSIYAFCCLFCS
LPLLGLGEHQQYCPGSWCFIRMRSAQPGGCAFSLAYASLMALLVTSIFFCNGSVTLSLYH
MYRQQRRHHGSFVPTSRAREDEVYHLILLALMTVIMAVCSLPLMIRGFTQAIAPDSREMG
DLLAFRFNAFNPILDPWVFILFRKAVFQRLKFWLCCLCARSVHGDLQAPLSRPASGRRDP
PAPTSLQAKEGSWVPLSSWGTGQVAPLTAVPLTGGDGCSVGMPSKSEAIAACSLC
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BDBM85181
n/a
NameBDBM85181
Synonyms:BERAPROST | CAS_2352 | NSC_2352
TypeSmall organic molecule
Emp. Form.C24H30O5
Mol. Mass.398.492
SMILESCC#CCC(C)C(O)C=CC1C(O)CC2Oc3c(cccc3CCCC(O)=O)C12 |w:8.7|
Structure
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