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TargetNorepinephrine transporter
LigandBDBM50005536
Substrate/Competitorn/a
Ki 0.47±n/a nM
CommentsPDSP_1164
Citation Owens MJMorgan WNPlott SJNemeroff CB Neurotransmitter receptor and transporter binding profile of antidepressants and their metabolites. J Pharmacol Exp Ther 283:1305-22 (1997) [PubMed]  Article
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Norepinephrine transporter
Name:Norepinephrine transporter
Synonyms:n/a
Type:Enzyme Catalytic Domain
Mol. Mass.:2082.45
Organism:RAT
Description:Norepinephrine transporter 0 RAT::Q9JIA2
Residue:19
Sequence:
MLLARMKPQVQPELGGADQ
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  Blast E-value cutoff:
BDBM50005536
n/a
NameBDBM50005536
Synonyms:42-548 | 5-(4-Chloro-phenyl)-2,5-dihydro-3H-imidazo[2,1-a]isoindol-5-ol | 5-(4-chlorophenyl)-3,5-dihydro-2H-imidazo[2,1-a]isoindol-5-ol | 5-Thiophen-2-yl-2,3,5,6-tetrahydro-imidazo[2,1-a]isoquinolin-5-ol | CHEMBL781 | MAZINDOL | Mazanor | Sanorex | mazindole
TypeSmall organic molecule
Emp. Form.C16H13ClN2O
Mol. Mass.284.74
SMILESOC1(N2CCN=C2c2ccccc12)c1ccc(Cl)cc1 |c:5|
Structure
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