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TargetSSTR2
LigandBDBM82470
Substrate/Competitorn/a
Ki 1.47±n/a nM
CommentsPDSP_373
Citation Meyerhof W The elucidation of somatostatin receptor functions: a current view. Rev Physiol Biochem Pharmacol 133:55-108 (1998) [PubMed]  Article
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SSTR2
Name:Somatostatin receptor
Synonyms:SOMATOSTATIN SST2 | SRIF-1 | SS2R | Somatostatin receptor 2 | Somatostatin receptor type 2
Type:Enzyme Catalytic Domain
Mol. Mass.:41212.21
Organism:RAT
Description:SOMATOSTATIN SST2 SSTR2 RAT::P30680
Residue:369
Sequence:
MELTSEQFNGSQVWIPSPFDLNGSLGPSNGSNQTEPYYDMTSNAVLTFIYFVVCVVGLCG
NTLVIYVILRYAKMKTITNIYILNLAIADELFMLGLPFLAMQVALVHWPFGKAICRVVMT
VDGINQFTSIFCLTVMSIDRYLAVVHPIKSAKWRRPRTAKMINVAVWGVSLLVILPIMIY
AGLRSNQWGRSSCTINWPGESGAWYTGFIIYAFILGFLVPLTIICLCYLFIIIKVKSSGI
RVGSSKRKKSEKKVTRMVSIVVAVFIFCWLPFYIFNVSSVSVAISPTPALKGMFDFVVIL
TYANSCANPILYAFLSDNFKKSFQNVLCLVKVSGAEDGERSDSKQDKSRLNETTETQRTL
LNGDLQTSI
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  Blast E-value cutoff:
BDBM82470
n/a
NameBDBM82470
Synonyms:3-(2-Naphtyl)-D-Ala-L-Cys(1)-L-Tyr-D-Trp-L-Lys-L-Val-L-Cys(1)-L-Thr-NH2 | BIM 23014 | BIM-23014 | LANREOTIDE
TypeSmall organic molecule
Emp. Form.C54H69N11O10S2
Mol. Mass.1096.323
SMILESCC(C)[C@@H]1NC(=O)[C@H](CCCCN)NC(=O)[C@@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](Cc2ccc(O)cc2)NC(=O)[C@H](CSSC[C@H](NC1=O)C(=O)N[C@@H]([C@@H](C)O)C(N)=O)NC(=O)[C@H](N)Cc1ccc2ccccc2c1
Structure
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