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TargetMelatonin receptor
LigandBDBM29611
Substrate/Competitorn/a
Ki 0.01±n/a nM
CommentsPDSP_1192
Citation Beresford IJBrowning CStarkey SJBrown JFoord SMCoughlan JNorth PCDubocovich MLHagan RM GR196429: a nonindolic agonist at high-affinity melatonin receptors. J Pharmacol Exp Ther 285:1239-45 (1998) [PubMed]
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Melatonin receptor
Name:Melatonin receptor
Synonyms:MTNR1A | MTNR1A protein | Mel-1A-R | Mel1a melatonin receptor | Melatonin 1A | Melatonin receptor 1A | Melatonin receptor type 1 (MT1) | Melatonin receptor type 1A
Type:Enzyme
Mol. Mass.:39392.94
Organism:Homo sapiens (Human)
Description:P48039
Residue:350
Sequence:
MQGNGSALPNASQPVLRGDGARPSWLASALACVLIFTIVVDILGNLLVILSVYRNKKLRN
AGNIFVVSLAVADLVVAIYPYPLVLMSIFNNGWNLGYLHCQVSGFLMGLSVIGSIFNITG
IAINRYCYICHSLKYDKLYSSKNSLCYVLLIWLLTLAAVLPNLRAGTLQYDPRIYSCTFA
QSVSSAYTIAVVVFHFLVPMIIVIFCYLRIWILVLQVRQRVKPDRKPKLKPQDFRNFVTM
FVVFVLFAICWAPLNFIGLAVASDPASMVPRIPEWLFVASYYMAYFNSCLNAIIYGLLNQ
NFRKEYRRIIVSLCTARVFFVDSSNDVADRVKWKPSPLMTNNNVVKVDSV
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  Blast E-value cutoff:
BDBM29611
n/a
NameBDBM29611
Synonyms:2-Iodomelatonin | CHEMBL289233 | Melatonin,2-Iodo
TypeSmall organic molecule
Emp. Form.C13H15IN2O2
Mol. Mass.358.1749
SMILESCOc1ccc2[nH]c(I)c(CCNC(C)=O)c2c1
Structure
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